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methyl 1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
1-{5-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
3-(morpholine-4-carbonyl)-N-[2-(1,3-thiazol-2-yl)ethyl]benzene-1-sulfonamide
6-[(4-methoxy-2,3-dimethylphenyl)methyl]-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
1-(4-fluorophenyl)-4-[7-(pyridin-3-yl)-9-[2-(thiophen-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butane-1,4-dione
[(3R,4R)-4-[(dimethylamino)methyl]-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)pyrrolidin-3-yl]methanol
5-{3-[2-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-oxopropyl}-5-[(4-methoxyphenyl)methyl]pyrrolidin-2-one
N-({8-[(4-methoxy-3-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)pyridine-3-carboxamide
N-[(2R,3R)-2-ethoxy-1'-[3-(1,2-oxazinan-2-yl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-4-(pyrrolidin-1-ylmethyl)benzamide
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(naphthalen-2-yl)ethan-1-one
N-methyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(pyrimidin-4-ylmethyl)piperidine-3-carboxamide
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-1-(3-propoxypiperidin-1-yl)propan-1-one
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-[3-(dimethylamino)-2,2-dimethylpropyl]-4-(piperidin-3-yl)benzamide
5-{3-[3-(2-chlorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-(thiophen-2-ylmethyl)pyrrolidin-2-one
N-[3-(3-methylphenyl)phenyl]-1-(6-methylpyridine-2-carbonyl)piperidine-3-carboxamide
3-amino-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)butanamide
(3R,4S)-1-(6-chloro-8-methylquinolin-4-yl)-4-cyclopropylpyrrolidin-3-amine
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl][(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
1-(4-methanesulfonylbenzoyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]-4-phenyl-1,2,3,6-tetrahydropyridine
(2E)-1-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(pyridin-3-yl)prop-2-en-1-one
2-(phenylsulfanyl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
1-tert-butyl-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyrrolidin-2-one
1-(2-methanesulfonylethyl)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazine
(1S,5R)-3-benzyl-6-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-{5-[(3-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(morpholin-4-yl)propan-1-one
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(2-methylphenyl)-1,3-benzoxazol-6-yl]acetamide
1-[(4-fluorophenyl)methyl]-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-1,4-diazepane
N-({7-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
8-[(3,5-dimethoxyphenyl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[(2,5-difluorophenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(3-methoxyphenyl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
1-(1-{1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperidin-4-yl}ethyl)-4-methylpiperazine
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
5-(5-fluoro-2-methylphenyl)pyrazin-2-amine
N-[1-(7-{[5-(2-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-methylpropanamide
2-[(2-fluorophenyl)methyl]-N-methyl-N-(pyridin-3-ylmethyl)-1,3-benzoxazole-6-carboxamide
2-methoxy-N-[3-(4-{[1-(1,3-thiazol-5-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]benzamide
N-[(2,6-difluorophenyl)methyl]-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-4-carboxamide
2-phenyl-N-(1-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
1-(4-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
2-[4-(1-ethylpiperidine-3-carbonyl)piperazin-1-yl]-N-(pyridin-3-yl)acetamide
1-ethyl-6-methyl-N-[3-(methylamino)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{4-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[6-(dimethylamino)pyrazin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
ethyl 4-(3-phenylpropyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxylate