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6,7-dimethoxy-2-(5-methoxy-3-methyl-1H-indole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline
N-tert-butyl-2-{4-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-1-yl}acetamide
4-[(2S,4R)-1-(adamantan-2-yl)-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
1-({4-[(3,4-dimethylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-4-ol
N-benzyl-3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}propanamide
1-tert-butyl-4-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}pyrrolidin-2-one
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[3-(piperidin-1-yl)propyl]acetamide
1-(4-methylquinazolin-2-yl)-N-{[2-(trifluoromethoxy)phenyl]methyl}piperidine-4-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-2-one
N-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-difluorobenzamide
5-(4-fluorophenyl)-N-[2-(morpholin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(diethylamino)propanamide
1-(3-chlorophenyl)-4-(2-methoxyacetyl)-5-methylpiperazin-2-one
ethyl 4-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-3-yl]piperazine-1-carboxylate
(2E)-3-(3-fluorophenyl)-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]prop-2-enamide
8-chloro-2-{[methyl({[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}quinolin-4-ol
9-[(6-hydroxynaphthalen-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-ethyl-1-methyl-3-({1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pent-2-yn-1-yl)pyrrolidin-3-yl]-1H-indole-5-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N-{1-[7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclopropanecarboxamide
5-ethyl-2-(3-phenylpiperazin-1-yl)pyrimidine
N-(2-{[(3-methylphenyl)methyl]carbamoyl}phenyl)pyrrolidine-3-carboxamide
1-methyl-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
3-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(3-methoxypropyl)-N-methylacetamide
2-methyl-5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyrazine
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-2-(naphthalen-2-yloxy)propanamide
6-(2-cyclohexylacetyl)-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
N-methyl-N-(1-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidin-4-yl}-2-phenylethyl)thiophene-3-carboxamide
1-methyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
4-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}thiomorpholine
4-{3-[(methylsulfanyl)methyl]piperidin-1-yl}pyrimidine-5-carboxylic acid
3-{2-oxo-2-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethyl}-1,3-oxazolidin-2-one
N-(1,3-benzoxazol-2-ylmethyl)-5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
N-(2-fluoro-4-methylphenyl)-2-{[1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]formamido}acetamide
3-methoxy-N-(1-{7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]-1-(piperidin-1-yl)propan-1-one
1-methyl-2-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}-1H-indole
2-[2-(4-methoxy-4-phenylpiperidin-1-yl)-2-oxoethyl]-2-azaspiro[4.4]nonan-3-one
4-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl]-1H-pyrrole-2-carbonitrile
4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]-1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidine
1-[2-(3-aminopyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
N-(3-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}phenyl)acetamide
8-(4-hydroxybutan-2-yl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
2-(cyclohex-1-en-1-yl)-1-[3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]piperidin-1-yl]ethan-1-one