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(1R,5S)-6-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-6-azabicyclo[3.2.1]octane
2-(3-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
1-[2-(piperidin-2-yl)ethyl]-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyloxan-4-amine
N-[1-(4-{cyclopropyl[(trimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]oxolane-3-carboxamide
N-(furan-2-ylmethyl)-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methylbenzamide
1-(2-methoxyphenyl)-4-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-pyrazole
N3-[(4-methoxyphenyl)methyl]-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(3-methoxyphenyl)-1-{1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}ethyl]-N,3-dimethylbutanamide
{4-[(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}pyrrolidin-3-yl)methyl]phenyl}methanol
5-(2-hydroxy-4-methylpentanoyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-ethanesulfonamido-1-methyl-2-phenyl-N-(pyridin-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
1-(4,6-dimethylquinazolin-2-yl)-N-(2-methoxyethyl)-N-methylpiperidine-4-carboxamide
(4aR,7aS)-1-methyl-4-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-N-[2-(1H-imidazol-4-yl)ethyl]-1-methyl-4-(naphthalene-1-amido)pyrrolidine-2-carboxamide
4-(1H-indol-6-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(azepane-1-carbonyl)-1-ethyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(2R,3R)-1'-cyclohexanecarbonyl-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
methyl N-{2-[2-butyl-4-(4-chlorophenyl)-5-oxopiperazin-1-yl]-2-oxoethyl}carbamate
8-methyl-2-propyl-N-[2-(pyridin-4-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
(4aR,7aS)-1-ethyl-4-[(4-methoxypiperidin-1-yl)sulfonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-(2,5-dimethoxyphenyl)propanamide
6-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}piperazin-2-one
N-(dicyclopropylmethyl)-3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
1-{4-[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-4-oxobutyl}pyrrolidin-2-one
4-(3-acetylphenyl)-N-propylbenzamide
(benzylsulfamoyl)[2-(7-methyl-1H-indol-3-yl)ethyl]amine
5-methoxy-2-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1,4-dihydropyridin-4-one
1-{3-[3-(azetidin-1-ylmethyl)phenoxy]-2-hydroxypropyl}piperidin-4-ol
N-[1-({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)piperidin-4-yl]acetamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[(2,4-difluorophenyl)methyl]propanamide
2-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-5,7-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
(3-{2-ethyl-3H-imidazo[4,5-b]pyridin-6-yl}phenyl)methanol
2-(1,3-dimethyl-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-yl)pyridine
ethyl 4-[(2-chlorophenyl)methyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidine-4-carboxylate
4-[1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)piperidin-3-yl]pyrimidine
6-[(diethylamino)methyl]-N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
1,5-dimethyl-4-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-{5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carbonyl}-4-propylpiperazine
N'-(3-chlorophenyl)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]pentanediamide
3-(1H-1,3-benzodiazol-2-yl)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
4-cyclopentyl-2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidine
2-(1,3-dimethyl-4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-yl)pyridine
10-methoxy-5-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-(3-hydroxy-2,2-dimethylpropyl)-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
1-(dimethylamino)-2-{4-[3-(5-methylfuran-2-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
5-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-(furan-2-ylmethyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide