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(4aS,8aS)-4a-hydroxy-N-(3-methyl-1,2,4-thiadiazol-5-yl)-decahydroisoquinoline-2-carboxamide
4-(3-methoxypyridin-2-yl)phenol
[(3R,5R)-5-(pyrrolidin-1-ylmethyl)-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)piperidin-3-yl]methanol
(2R,6R)-10-methoxy-4-[3-(methylcarbamoyl)pyridin-2-yl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-(4-methoxyphenyl)-3-phenylpropanamide
4-{[5-(3,5-dimethyl-1-benzofuran-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methylpiperidine
N-methyl-5-oxo-1-(pyridin-3-ylmethyl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)pyrrolidine-3-carboxamide
7-chloro-3-methyl-2-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-indole
N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-phenoxyacetamide
1-(5-methyl-1H-pyrazole-3-carbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
methyl 8-[(5-ethylfuran-2-yl)methyl]-1-(3-methylbutoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-4-methylpiperazine-1-carboxamide
(3S,4R)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(hydroxymethyl)piperidin-3-ol
methyl (2R,4S)-4-hydroxy-1-(3-methoxybenzoyl)piperidine-2-carboxylate
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-1-[4-(2-ethoxyphenyl)piperazin-1-yl]ethan-1-one
3-({1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}oxy)pyridine
2-ethoxy-4-({[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenol
N-[(4-phenyloxan-4-yl)methyl]-6-(5-propyl-1,2-oxazole-3-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
5-{[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2,2-dimethyl-1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
2-methylpropyl 2-(phenylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
3-ethyl-1-[4-(1H-imidazol-1-yl)phenyl]-3-(2-methoxyethyl)urea
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-6-methylimidazo[1,2-a]pyridine-2-carboxamide
1-(3-benzyl-1H-1,2,4-triazol-5-yl)cyclopropane-1-carboxamide
N-[2-({2-methylimidazo[1,2-a]pyrimidin-3-yl}formamido)ethyl]pyridine-3-carboxamide
benzyl (1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-(pyrazin-2-yl)acetamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-phenylcyclopropane-1-carboxamide
3-{2-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
8-chloro-2-{[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}-1,4-dihydroquinolin-4-one
1-(benzenesulfonyl)-N-(4-methoxy-4-methylpentan-2-yl)piperidin-4-amine
1-[(4-methoxyphenyl)methyl]-5-[3-(trifluoromethyl)-1H-pyrazol-5-yl]-1H-1,2,4-triazole
N-{1-[1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide
N-(2-methoxyethyl)-1,5,6-trimethyl-2-oxo-N-(thiophen-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
5-methyl-N-[2-(pyridin-2-yl)ethyl]-6-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-[(2,5-difluorophenyl)methyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
7-chloro-4-(4,4-difluoropiperidine-1-carbonyl)-2-methylquinoline
2-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
2-[({5-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
1-cycloheptyl-N-methyl-6-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
1-[2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-N,N-dimethylpyrrolidin-3-amine
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-ethyl-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}pyridine-3-carboxylic acid
N-{3-[2-(isoquinolin-5-yl)-1H-imidazol-1-yl]phenyl}acetamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[2-(methylsulfanyl)ethyl]acetamide
1-(4-{1-azabicyclo[3.2.1]octan-5-yloxy}-3-methoxyphenyl)ethan-1-one
1-ethyl-3-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}piperidine
6-methoxy-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-4-amine
N-tert-butyl-2-(5,6-dimethylpyrimidin-4-yl)benzene-1-sulfonamide
methyl (4aR,7aS)-4-[(2,5-dimethoxyphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate