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3-{2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}-4-(propan-2-yl)piperazin-2-one
2-{[methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl})amino]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
5-[1-(3-cyclohexylpropanoyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
(2,2-dimethylpropyl)(methyl)({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amine
2-(morpholin-4-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}pyrimidine-5-carboxamide
1-(3,3-diphenylpiperidin-1-yl)-3-methoxypropan-1-one
4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-N,6-dimethylpyrimidin-2-amine
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[(2-methylpropyl)amino]methyl}piperidin-2-one
N-[(3R,4R)-1-{[4-(difluoromethoxy)phenyl]methyl}-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
[(4-fluorophenyl)methyl](methyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-{2-[4-(4-chlorophenyl)piperazin-1-yl]-2-oxoethyl}-1-cyclopropyl-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-(dimethylamino)-2-(2-fluorophenyl)ethan-1-one
ethyl 1-[3-(methylsulfanyl)propanoyl]-3-(2-phenylethyl)piperidine-3-carboxylate
2-{2-[4-(2,3-dichlorophenyl)-1H-1,2,3-triazol-1-yl]ethyl}-6-methyl-3,4-dihydropyrimidin-4-one
methyl 2-{[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidin-2-yl]formamido}acetate
2-methyl-1-{2-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-indole
2-(2H-1,2,3-benzotriazol-2-yl)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)acetamide
methyl(thiophen-2-ylmethyl){[3-(2-{4-[4-(trifluoromethyl)benzoyl]piperazin-1-yl}ethoxy)phenyl]methyl}amine
2-[5-(oxolan-2-yl)thiophen-2-yl]-1H-1,3-benzodiazole-6-carboxylic acid
N-cyclopentyl-N-{[3,5-dimethoxy-4-(oxolan-2-ylmethoxy)phenyl]methyl}-3-fluorobenzamide
4-(2-methyl-1H-imidazol-1-yl)-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidine-4-carboxylic acid
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-(2-oxopyrrolidin-1-yl)propanamide
3-[(4-fluorophenyl)methyl]-5-methyl-5-[1-(pyridine-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
(2S,5R)-2,5-dimethyl-1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
1-(2-methylpropyl)-8-(2-phenylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-6-propyl-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-2-(6-methoxynaphthalen-2-yl)morpholine
3-(cyclopropylmethyl)-5-(2-ethyl-4-fluorophenoxymethyl)-1,2,4-oxadiazole
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol
2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
N-[1-(1,3-thiazol-2-yl)ethyl]-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
7-(3-chlorophenyl)-4-[(1R,2S)-2-propylcyclopropanecarbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(5S,9aS,9bS)-5-(6-methoxy-2H-chromen-3-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[1-(3-methoxyphenyl)ethyl]-N-methylpropanamide
1-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)azepan-2-one
5-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]quinoxaline
4-ethyl-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
2-[1-({1-[2-(propan-2-yl)pyrimidine-5-carbonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
1-(2-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
N-(1-{1-[2-(4-chlorophenoxy)acetyl]piperidin-4-yl}-2-(2,4-difluorophenyl)ethyl)-N-methylpropanamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]propanamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-methanesulfonyl-2-methylpyrimidin-4-amine
1-methyl-4-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]piperidin-4-ol
methyl 4-{2-amino-3-cyano-5H-indeno[1,2-b]pyridin-4-yl}-1H-pyrazole-3-carboxylate
1-methanesulfonyl-4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-1H-pyrazole
1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-(3-phenylpropyl)-1,4-diazepane
2-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1-methylazepane