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2-[4-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
3-chloro-N-[(3S)-2-oxoazepan-3-yl]-N-({4-[3-(pyridin-3-yl)propoxy]phenyl}methyl)benzamide
1-[4-(8-methoxy-4-methylquinolin-2-yl)piperazin-1-yl]ethan-1-one
N-ethyl-2-{2-methylimidazo[1,2-a]pyridin-3-yl}-N-[2-(3-methylphenoxy)ethyl]acetamide
N-(2-{[(3R,5S)-5-(3-fluorophenoxymethyl)piperidin-3-yl]formamido}ethyl)acetamide
2-(1H-indol-3-yl)-1-(4-{2-[(3-methoxyphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)ethan-1-one
3-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-9-methoxy-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(2R)-N-[(4-methoxyphenyl)methyl]-2-methyl-N-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
4-[(4-fluorophenyl)methyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
N-ethyl-N-methyl-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-[1-(1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
(2S,3S)-2-amino-1-{4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-3-methylpentan-1-one
2-(2-{1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
1-(3,5-dimethoxyphenyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
3-[4-(4-amino-6,7-dimethoxyquinazolin-2-yl)phenyl]propanoic acid
N-cyclopropyl-1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
3-{3-[4-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}pyridin-1-ium-1-olate
5-benzamido-1-cyclopentyl-N-(3-ethoxypropyl)-1H-1,3-benzodiazole-7-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
2-(methylamino)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1,3-thiazole-4-carboxamide
1-[4-(3-chlorophenyl)piperazin-1-yl]-3-(3-methylpiperidin-1-yl)propan-1-one
3-ethyl-6-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-3H-imidazo[4,5-b]pyridin-2-amine
(5-{[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]methyl}furan-2-yl)methanol
5-(2-chlorophenyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]furan-2-carboxamide
1-(3-{[(dimethylsulfamoyl)amino]methyl}piperidin-1-yl)-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
1-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-N,N-diethylpiperidine-3-carboxamide
2-(2-{[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]amino}ethyl)-6-methyl-3,4-dihydropyrimidin-4-one
N-(1-{1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]piperidin-4-yl}-2-(2-methylphenyl)ethyl)-N-methyl-2-(1H-pyrazol-1-yl)acetamide
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
4-(2-methyl-1H-imidazol-1-yl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidine-4-carboxylic acid
{3-[(2-fluorophenyl)methyl]-1-(3-methoxypyrazin-2-yl)piperidin-3-yl}methanol
1-[(diethylcarbamoyl)methyl]-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-(dimethylamino)-2-(4-fluorophenyl)-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
8-(furan-3-carbonyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1R,5R)-6-(cyclobutylmethyl)-3-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(pentan-3-yl)-N-(2-phenylethyl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
2-{2-[5-(pentan-2-yl)-4-phenyl-1H-imidazol-1-yl]ethoxy}ethan-1-ol
methyl 6-[2-(cyclohex-1-en-1-yl)acetyl]-2-[(4-fluorophenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
2-methoxy-N-[(2R,3R)-1'-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-(1-{1-[2-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
5-(2-methylpropyl)-1'-(pyrazine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
1-[(2S)-2-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrrolidin-1-yl]ethan-1-one
4-({[3-(4-fluorophenoxy)propyl](methyl)amino}methyl)-N-methylbenzene-1-sulfonamide
(4-{[(3-methoxypyrazin-2-yl)(methyl)amino]methyl}oxan-4-yl)methanol
4-{3-cyclopropyl-5-[2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)ethyl]-1H-1,2,4-triazol-1-yl}-3-methylpyridine
(1S,5R)-3-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[4-({[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}methyl)phenyl]prop-2-yn-1-ol