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2-(3,4-dimethoxyphenyl)-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
N-[2-methyl-2-(morpholin-4-yl)propyl]-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
3-(4-{[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)phenol
8-[(2,6-difluorophenyl)methyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
(3aR,6aR)-2-methanesulfonyl-5-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(3-chloro-4-hydroxyphenyl)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}ethan-1-one
1-cyclohexyl-6-(pyridin-2-ylmethoxy)-4-[2-(pyridin-4-ylsulfanyl)acetyl]-1,4-diazepan-2-one
4-(4-ethoxy-3-methylphenyl)-N-methyl-N-(1-methylpiperidin-4-yl)butanamide
2-methoxy-N-{1-[1-(oxan-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-{4-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-1-cyclopentylpiperazin-2-yl}ethan-1-ol
1-(cyclopropylmethyl)-3-(2-methylquinolin-5-yl)-6-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(3-chloro-4-methoxyphenyl)-6-(3-phenylprop-2-ynoyl)-6-azaspiro[2.5]octane-1-carboxamide
5-methyl-2-[2-({2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]pyrimidin-4-amine
N-(1-{7-[4-(furan-2-yl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
2-ethyl-4-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}morpholine
4-[(3-phenylphenyl)methyl]-4H-1,2,4-triazole
2-[1-(cyclohexylmethyl)-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
N-{[2-(difluoromethoxy)phenyl]methyl}-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(2R,3R)-3-[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
9-ethyl-3-{[1-(4-methyl-1,4-diazepane-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]methyl}-9H-carbazole
3-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
3-({2-[4-(propan-2-yl)-1,3-thiazol-2-yl]-1H-imidazol-1-yl}methyl)-1λ6-thiolane-1,1-dione
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(2R,3R)-1'-(3-methoxybenzoyl)-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
2-amino-4-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-(furan-2-yl)pyridine-3-carbonitrile
N-[7-(4-formylpiperazine-1-carbonyl)-1-methyl-2-phenyl-1H-1,3-benzodiazol-5-yl]ethane-1-sulfonamide
5-butyl-4-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-1-(3-methylphenyl)piperazin-2-one
1-[4-({[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
6-[(2-chloro-4,5-dimethoxyphenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-[3-(trifluoromethyl)phenyl]piperazine
(3S,4S)-1-(5-chloro-2-fluorobenzoyl)-4-methylpiperidine-3,4-diol
3-amino-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-1H-1,2,4-triazole-5-carboxamide
3-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}pyridin-2-ol
2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-imidazole
2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-(oxolan-3-yl)acetamide
N-(4-chloro-2-methylphenyl)-4-[(1-methylpiperidin-3-yl)methyl]piperazine-1-carboxamide
1-[4-(3-fluorophenoxy)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
N-({7-[(3-ethoxy-4-hydroxyphenyl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
1-[2-methoxy-5-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-(4-{[4-(3-methylbutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-ol
6-[(3-methoxyphenyl)methoxy]-4-(1H-pyrazol-3-ylmethyl)-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
N-[2-(4-ethylmorpholin-2-yl)ethyl]-3-methylthiophene-2-carboxamide
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-3,5-difluoropyridine
1-(2H-1,3-benzodioxol-4-ylmethyl)-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
8-cyclopentyl-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione