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4-(4-butoxyphenyl)-7-(2-oxoimidazolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
(4aS,8aR)-6-(3-chlorobenzoyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
2-[3-(1H-imidazol-1-yl)propyl]-5-(3-methoxypiperidine-1-carbonyl)-2,3-dihydro-1H-isoindol-1-one
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)cyclohexyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[1-(5-methyl-1,3,4-oxadiazol-2-yl)azetidin-3-yl]piperidine
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-(3-phenylpropyl)piperazin-2-one
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]acetamide
6-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-ylmethyl]-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]piperidine
(1S,5R)-3-(2H-1,3-benzodioxole-5-carbonyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(cyclohexylmethyl)-1H-pyrazol-5-yl]-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carboxamide
3-[5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
1-(3-methoxy-4-methylphenyl)-3-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
3-(2-amino-1,3-thiazol-4-yl)-N-[3-(morpholin-4-yl)propyl]propanamide
4-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
N-({3-methyl-7-[2-(1H-pyrazol-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
{[3-(2-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-2-yl}ethoxy)phenyl]methyl}(methyl)(quinolin-8-ylmethyl)amine
(2S,4R)-4-(dimethylamino)-1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrrolidine-2-carboxylic acid
3-(1H-1,3-benzodiazol-2-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]propan-1-one
(4aS,8aR)-6-(1,2-oxazole-3-carbonyl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-methyl-1H-indole-2-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-(2-methyl-4-phenylpiperazin-1-yl)ethan-1-one
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-6-(propan-2-yl)pyridazin-3-amine
2-(1,4-dimethylpiperazin-2-yl)-N-(3-hydroxypropyl)-N-(naphthalen-1-ylmethyl)acetamide
1-[1-(cyclopropanesulfonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
butyl(furan-2-ylmethyl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
3-(1-phenylethyl)-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}-1,2-oxazole-5-carboxamide
(1R,7S)-3-(2-ethoxyethyl)-6-(4-methylpiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(cyclohex-1-en-1-yl)acetamide
2-({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-amine
1-ethyl-4-[({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-1H-pyrrole-2-carbonitrile
3-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]-1λ6-thiolane-1,1-dione
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[(3R,4S)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-{4-[(4-ethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-3-methylbutan-1-ol
2-[methyl(pyridin-3-ylmethyl)amino]-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethan-1-one
2-[(2-methoxyethyl)(methyl)amino]-2-(naphthalen-2-yl)acetic acid
3-phenyl-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperazine
2,4-dimethyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-1,3-oxazole-5-carboxamide
[(3R,4R)-1-(2-chloro-6-fluorobenzoyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
4-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-1,2-dimethylpiperazine
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
5-({3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)pyrimidine
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]propanamide