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2-(3-methoxyphenyl)-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
N-{[7-(2,2-dimethylpropanoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
[4-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)oxan-4-yl]methanol
1-({1-[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}methyl)pyrrolidin-2-one
4-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
8-[(1R,9aR)-octahydro-1H-quinolizine-1-carbonyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4R)-1-[(2,5-difluorophenyl)methyl]-N-(furan-3-ylmethyl)-4-[(4-methoxyphenyl)sulfanyl]-N-methylpyrrolidine-2-carboxamide
N-(2-methoxyethyl)-2-[(propan-2-yl)amino]-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
N-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-methoxyethyl)propanamide
2-(3-oxo-9-{spiro[2.3]hexane-1-carbonyl}-2,9-diazaspiro[5.5]undecan-2-yl)acetic acid
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(3-methylpyridin-2-yl)piperazine
4-methoxy-N-[2-(7-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
2-{1,4-bis[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(2-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}phenoxy)ethan-1-ol
3-ethyl-1-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-3-ol
N-[(2R,3R)-1'-[(2,6-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
(2-ethoxy-5-{[propyl(pyridin-3-ylmethyl)amino]methyl}phenyl)methanol
(1R,5S,6R)-N-[2-(4-ethoxyphenyl)ethyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
1-methyl-6-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-1H-indole
3-(piperidin-1-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
6-(3-chlorophenyl)-N-methyl-N-(pyridin-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-1-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}propan-1-one
(1R,5R)-6-[(3-chloro-4-fluorophenyl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-methyl-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)imidazo[2,1-b][1,3]thiazole-5-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]pyridine-4-carbonitrile
3-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]-N-(1,3-thiazol-2-yl)propanamide
N3-benzyl-1-cyclopropyl-N5-[(2,6-difluoro-3-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[9-(4-methoxy-3-methylbenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
(1R,5S,6S)-N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexane-3-carboxamide
1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
7-fluoro-3-{[(2-methylpropyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}-1,2-dihydroquinolin-2-one
N-[1-(1H-indol-5-yl)ethyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)benzamide
5-{3-[3-(methoxymethyl)piperidin-1-yl]-3-oxopropyl}-5-[(4-methoxynaphthalen-1-yl)methyl]pyrrolidin-2-one
9-methoxy-7-(6-methoxypyridazin-3-yl)-4-(1-phenylcyclohexanecarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-({7-[3-(3-fluorophenyl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
(3E)-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pent-3-enamide
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[2-(pyridin-2-yl)ethyl]acetamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-chloro-6-fluoro-3-methylbenzamide
1-(2-aminoethyl)-N-[2-(cyclohexylsulfanyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-9-methoxy-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
5-[1-(3-chloro-4-fluorobenzoyl)piperidin-4-yl]-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
(2R,3R,6R)-3-(4-fluorophenyl)-5-(4-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-benzyl-3-propyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-[3-(3-chlorophenyl)phenyl]-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-amine