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1-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
1-[2-({[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}amino)pyrimidin-4-yl]piperidin-3-ol
N-[(2-ethoxyphenyl)methyl]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
4-[(1-butyl-1H-1,3-benzodiazol-2-yl)methyl]-1λ6-thiomorpholine-1,1-dione
cyclopentyl 4-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}amino)benzoate
(3S,4S)-1-(2-methyl-6-propylpyrimidin-4-yl)-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
N-cyclopentyl-N'-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N'-(pyridin-3-ylmethyl)butanediamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-3-phenylpropan-1-one
N-(1-{7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylbenzamide
5-amino-4-chloro-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1H-pyrazole-3-carboxamide
3-(3-fluoro-4-methoxybenzoyl)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidine
8-[(3-ethoxy-4-methoxyphenyl)methyl]-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2E)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-phenylprop-2-enamide
2-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}ethan-1-ol
(3R,4R)-3-cyclobutyl-1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-4-methylpyrrolidin-3-ol
2-amino-6-methyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]pyrimidine-4-carboxamide
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4,4,4-trifluorobutanamide
3-[2-(azonan-1-yl)-2-oxoethyl]-4-(2-phenylethyl)piperazin-2-one
2-[3-({[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)phenoxy]ethan-1-ol
2-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
6-(furan-2-yl)-2-(4-{[3-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-ethylbenzamide
4-{[2-(2-carboxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-oxo-2H-chromene-3-carboxamide
(3S,4S)-1-(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)piperidine-3,4-diol
1-(benzyloxy)-8-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-1,8-diazaspiro[4.5]decan-2-one
(5-tert-butyl-1-methyl-1H-1,2,4-triazol-3-yl)(phenyl)methanol
5-methyl-N-({1-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-3-yl}methyl)-1,2-oxazole-3-carboxamide
2-{2-methylimidazo[1,2-a]pyridin-3-yl}-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]acetamide
4-(2-methoxyethyl)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1,4-diazepan-5-one
1-(2-fluorophenyl)-N-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-amine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[5-(hydroxymethyl)furan-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-2,9-diazaspiro[5.5]undecan-3-one
N-cyclobutyl-3-{[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]sulfonyl}benzamide
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}amine
2-ethyl-N-[2-(2-methoxyphenyl)ethyl]-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
1-[3-(morpholine-4-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-phenylpropan-1-one
1-methyl-3-phenyl-8-[2-(propylsulfanyl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
2-amino-N-(2H-1,3-benzodioxol-5-ylmethyl)-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(4-methylphenyl)methyl]piperidine-3-carboxamide
N-[1-(1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-methylbutanamide
3-[(4-ethylphenyl)methyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
methyl 1-(benzyloxy)-8-[(4-fluorophenyl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
9-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-chloro-4-fluorophenoxy)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
2-{1-cyclopentyl-4-[(2-methoxynaphthalen-1-yl)methyl]piperazin-2-yl}ethan-1-ol