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(2S)-2-amino-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-(1H-imidazol-4-yl)propan-1-one
2-[4-fluoro-3-(hydroxymethyl)phenyl]-2-[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]acetic acid
ethyl 3-[(2-fluorophenyl)methyl]-1-[3-(1H-indol-3-yl)propanoyl]piperidine-3-carboxylate
(1R,5S,8R)-8-methoxy-3-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-3-azabicyclo[3.2.1]octane
ethyl 1-(2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperidine-4-carboxylate
4-(1H-indol-4-yl)-5,6,7-trimethoxy-1,2,3,4-tetrahydroquinolin-2-one
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyridine-3-carboxamide
6-[(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)methyl]pyridine-2-carboxylic acid
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(1,3-thiazol-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
6-{[3-(diethylcarbamoyl)piperidin-1-yl]methyl}-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{5-[(2E)-but-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-cyclopropylpropanamide
5-methyl-5-[1-(9-methyl-9H-carbazole-3-carbonyl)piperidin-4-yl]-3-(pyridin-4-ylmethyl)imidazolidine-2,4-dione
4-(azocan-1-yl)-5-methyl-N-[2-(propan-2-yloxy)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-(2-aminoethyl)-2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzamide
(2S)-2-acetamido-4-(methylsulfanyl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]butanamide
2-amino-4-cyclopentyl-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
1-(2-methoxyethyl)-3-(2-phenylethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-3-(2-methylpropyl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1,2-oxazole-5-carboxamide
5-[1-(furan-3-ylmethyl)pyrrolidin-2-yl]-N-[2-(pyridin-4-yl)ethyl]thiophene-2-carboxamide
9-methoxy-N-[(2-methoxyphenyl)methyl]-3-[(4-methyl-1H-imidazol-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-3-(pyridin-3-yl)propanamide
(3S,4S)-4-(naphthalen-2-yl)-1-(thiophene-2-carbonyl)piperidin-3-ol
2-{5-[(4-methanesulfonylphenyl)methyl]-3-methyl-1H-1,2,4-triazol-1-yl}pyridine
9-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1,3,5-trimethyl-1H-pyrazol-4-amine
2-{4-[(4-fluorophenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-methoxy-2-phenyl-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-[2-(dimethylsulfamoyl)ethyl]-4-(pyrrolidin-1-ylmethyl)benzamide
N-(2-methoxyethyl)-6-methyl-N-(pyridin-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-5-carboxamide
4-(2-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-2-yl}ethyl)phenol
5-(1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-2-yl)-3-phenyl-1,2,4-oxadiazole
3,5-difluoro-2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]pyridine
N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-[2-(4-methylphenoxy)ethyl]acetamide
ethyl 1-[(4-hydroxy-3-methoxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
(1s,4s)-4-({methyl[1-(pyridin-2-yl)propyl]amino}methyl)cyclohexan-1-amine
5-chloro-3-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-4-(3,3,3-trifluoropropyl)pyrimidine
1-(6-methoxy-4-methylquinazolin-2-yl)-N-[1-(thiophen-2-yl)propan-2-yl]piperidin-4-amine
2-amino-4-(3-chloro-5-fluoro-4-methoxyphenyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
3-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(3,4-dimethoxyphenyl)-1-(2,3-dimethyl-1H-indole-7-carbonyl)piperidin-3-amine
(1R,5R)-6-(2-methoxyethyl)-3-(3-methylthiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[2-(4-methoxyphenyl)ethyl]-3-(1,3,4-thiadiazol-2-yl)urea
[(3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](1H-imidazol-2-ylmethyl)methylamine
N-methyl-N-[2-(4-methylphenoxy)ethyl]-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
1-[1-(pyridin-2-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]but-3-en-1-one
3-(morpholine-4-carbonyl)-1-propyl-N-{[4-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
N-[2-(dimethylamino)ethyl]-5-(isoquinolin-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide