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3-(2-chlorophenyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]propanamide
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-3-methylpentanamide
2-(2-methylphenyl)-5-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)pyrimidine
2-[4-(2,2-dimethylpropyl)-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethylpyrrolidin-3-amine
9-[(2S)-2-amino-4-(methylsulfanyl)butanoyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
N-[2-(cyclohexylsulfanyl)ethyl]-4-methylpyrimidin-2-amine
1-(cyclohex-1-ene-1-carbonyl)-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
(3aS,6aR)-5-(1H-indol-3-ylmethyl)-3-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-ethylpiperazin-1-yl)acetamide
(3R,4R)-4-methyl-3-(propan-2-yl)-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)pyrrolidin-3-ol
2-{[4-(4-chlorophenyl)-5-(1-ethoxyethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(1H-imidazol-2-ylmethyl)(2-methylpropyl)(pyridin-2-ylmethyl)amine
4-(2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)piperazin-2-one
2-{2-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-4-phenyl-1,2-dihydrophthalazin-1-one
4-{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidine-4-carbonyl}morpholine
4-{3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
5-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
methyl 6-(piperidin-1-ylmethyl)-3-(thiophene-3-amido)thieno[2,3-b]pyridine-2-carboxylate
N-[5-({7-[(2-chloro-6-fluorophenyl)(hydroxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)thiophen-2-yl]acetamide
N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]-1-(propan-2-yl)piperidine-3-carboxamide
4-chloro-2-methoxy-N-[(1-methylpiperidin-3-yl)methyl]benzamide
ethyl 4-benzyl-1-(1H-indol-3-ylmethyl)piperidine-4-carboxylate
N-[(3S,4R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
4-[(1,1-dioxo-1λ6-thian-3-yl)methyl]-N-propylbenzamide
N-(furan-2-ylmethyl)-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
(1S,5R)-N-(3-chlorophenyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(furan-2-ylmethyl)-N-(2-phenylethyl)acetamide
4-methyl-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]benzene-1-sulfonamide
N-[1-(4-methanesulfonylphenyl)propyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
({1-[(1-hexylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)(methyl)amine
N-{2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}acetamide
2-(4-chloro-2-{[2-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)acetamide
N-(3,3-diphenylpropyl)-6-[(4R)-2-oxo-1,3-thiazolidine-4-carbonyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{1-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]piperidin-4-yl}acetamide
4-[(8-methoxy-2H-chromen-3-yl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
1-methyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-(piperidine-1-sulfonyl)piperidine-4-carboxylic acid
2-methyl-8-{2-[3-(methylsulfanyl)phenyl]acetyl}-2,8-diazaspiro[4.5]decan-3-one
(2R)-2-amino-1-{7-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}propan-1-one
4-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]thiomorpholine
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
3-{[4-(dimethylamino)oxan-4-yl]methyl}-1-[3-(3-methoxyphenyl)phenyl]urea
2-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-hydroxyethyl]phenol
N-[(2-chloropyridin-3-yl)methyl]-2-methoxy-N,4-dimethyl-1,3-thiazole-5-carboxamide
1-{1'-[(5-methylthiophen-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
5-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-amine