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3-({[(2-amino-1,3-thiazol-4-yl)methyl]amino}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
1-(6-methyl-2-phenylpyrimidin-4-yl)-N-(thiolan-3-yl)piperidin-4-amine
1-(4-methoxyphenyl)-N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)cyclopentane-1-carboxamide
7-fluoro-N,N-dimethyl-2-[2-(pyridin-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
2-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazine-1-carbonyl)pyridin-3-ol
1-{[3-(morpholin-4-yl)phenyl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
6-(naphthalene-1-carbonyl)-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
1-benzyl-8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(dicyclopropylmethyl)-2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
4-methoxy-3-{1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
(3aS,6aS)-2-benzyl-5-(1H-pyrazole-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-methyl-3-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-[2-(oxan-4-yl)ethyl]propanamide
N-(3-{5-methyl-4-[(3-phenylpropanamido)methyl]-1,3-oxazol-2-yl}phenyl)oxane-4-carboxamide
3-(1H-imidazol-4-ylmethyl)-4-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)piperazin-2-one
3-[2-(dimethylamino)ethyl]-8-(2-ethylbutyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(1-{[1-(furan-3-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]urea
(3S,4R)-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-3-methoxypiperidin-4-amine
1-cyclohexyl-N-(piperidin-4-yl)-N-(pyridin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(2E)-N-{[7-(3,4-difluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
[4-(2-phenoxyethyl)piperidin-4-yl]methanol
N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
8-(furan-3-ylmethyl)-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1,3-benzoxazol-2-ylmethyl)-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-cyclopropyl-1-[2-(3,4-dimethoxyphenyl)ethyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
(2S,4S)-1-(2,4-dimethylbenzoyl)-N-ethyl-4-(pent-4-enamido)pyrrolidine-2-carboxamide
1-[(6-chloropyridin-3-yl)methyl]-3-(2-methylpropyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(1,3-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[3-(4-{[2-(3-chlorophenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-3-methylbutanamide
1-methyl-5-[4-(methylsulfanyl)benzoyl]-N-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-1-cyclopentyl-3-(3-fluorophenyl)pyrrolidine-2,5-dione
2-butyl-8-(5-methoxyfuran-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{5-[1-(ethanesulfonyl)ethyl]-3-phenyl-1H-1,2,4-triazol-1-yl}-3-methylpyridine
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2-hydroxypropyl)-1H-pyrazole-3-carboxamide
N5,N5,N6-trimethyl-N6-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-(2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}ethyl)piperidin-4-ol
N-[1-(benzenesulfonyl)piperidin-4-yl]imidazo[1,2-a]pyrimidine-2-carboxamide
1-[(2-methoxyphenyl)methyl]-6-oxo-N-[2-(propan-2-yloxy)ethyl]piperidine-3-carboxamide
2-(3-{[(3-hydroxypropyl)(methyl)amino]methyl}phenyl)-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
4-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-2-methyl-1,3-oxazole
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(4,6-dimethylquinazolin-2-yl)-N-methylpiperidine-4-carboxamide
N-(2-{7-[(4-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
4-({2-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
3-chloro-4-fluoro-N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]benzamide
N,1,7-trimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H-indole-2-carboxamide
2-(2-methoxyphenoxy)-N-{[1-(pyridin-3-ylmethyl)piperidin-3-yl]methyl}acetamide
N-[3-(cyclohexyloxy)-2-hydroxypropyl]-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
6-methyl-2-oxo-N-[(1r,4r)-4-methoxycyclohexyl]-1,2-dihydropyridine-4-carboxamide
9-[(5-ethylpyridin-2-yl)methyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one