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methyl 1-(2-methylpropyl)-3-(2-phenylacetamido)-5-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3S,9aR)-8-[(2-fluoro-5-methylphenyl)methyl]-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(1-benzofuran-2-carbonyl)-6-(cyclopropylmethoxy)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-[3-(furan-2-yl)propyl]-7-(pyrimidin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-({[(5-chloro-2-methoxyphenyl)methyl](methyl)amino}methyl)pyridine-3-carboxylic acid
{5-[3-(morpholin-4-ylmethyl)phenyl]-2-propoxyphenyl}methanol
3-ethoxy-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-(1-benzofuran-2-yl)-1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-imidazole
[(3R,4R)-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-tert-butyl-2-({6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl}formamido)acetamide
1-[2-methoxy-5-({[2-(thiophen-2-yl)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)[3-(pyrrolidin-1-yl)butyl]amine
5-methyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-1,2-oxazole-4-sulfonamide
(1R,5S,6R,7S)-3-(2-aminoethyl)-6-[4-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]decan-4-one
3-(4-chlorobenzoyl)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
N-[(2R,3R)-2-(pyridin-2-ylmethoxy)-1'-(2,2,3,3-tetramethylcyclopropanecarbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-[3-(4-{[1-(2-chlorophenyl)ethyl]amino}piperidin-1-yl)phenyl]ethane-1-sulfonamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-1-[4-(3-methylpyridin-4-yl)piperazin-1-yl]propan-1-one
3-(1,3-benzothiazol-2-yl)-N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)propanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-2-ylmethyl)pyrrolidin-3-yl]-2-(methylamino)-1,3-thiazole-4-carboxamide
3-(1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}piperidin-3-yl)-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
[(2,3-dimethyl-1H-indol-5-yl)methyl](1-methoxypropan-2-yl)amine
N-{4-[1-(cyclopent-3-en-1-yl)-4-phenyl-1H-imidazol-5-yl]phenyl}acetamide
N-(2-chlorophenyl)-3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-(2-butoxy-5-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-(1-{[4-(benzyloxy)phenyl]methyl}piperidin-4-yl)-5-methylimidazolidine-2,4-dione
2-[(3,4-difluorophenyl)methyl]-8-(furan-3-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
5-methoxy-N,1,2-trimethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1H-indole-3-carboxamide
N-(1-methanesulfonylpiperidin-4-yl)-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-1-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
N-{2-[(2R,3R)-2-methoxy-3-(2-phenylacetamido)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-oxoethyl}acetamide
N,1-dimethyl-N-(2-{[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]oxy}hex-5-en-1-yl)piperidin-4-amine
3-[(4-fluorophenyl)methyl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
N-{1-[1-(2,5-dimethylbenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,3-dimethylbutanamide
N-[(3R,4S)-4-(propan-2-yl)-1-(1H-1,2,3-triazol-4-ylmethyl)pyrrolidin-3-yl]oxane-4-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}quinoxaline-6-carboxamide
4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1-phenylpiperazine-2-carboxylic acid
1-benzyl-8-[(2E)-3-phenylprop-2-en-1-yl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2-(pyridin-2-yl)acetamide
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(pent-2-yn-1-yl)piperidine
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
6-chloro-2-methyl-4-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}quinoline
N-(3-chlorophenyl)-3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
1-[6-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroquinolin-1-yl]ethan-1-one
4-fluoro-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]benzamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
N-[(3,5-difluorophenyl)methyl]-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide