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N-[(8-methoxyquinolin-5-yl)methyl]-N,1-dimethylazepane-2-carboxamide
(3R,4R)-1-cyclobutanecarbonyl-4-{[(3-phenyl-1H-pyrazol-5-yl)methyl]amino}pyrrolidin-3-ol
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,5-dimethylfuran-3-carboxamide
N-(1-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-2-carboxamide
4-methyl-N-{3-[2-(oxolan-3-yl)-1H-imidazol-1-yl]propyl}benzene-1-sulfonamide
1-[cyclohexyl(methyl)amino]-3-[3-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
5-(5-methylfuran-2-yl)-N-(oxan-4-ylmethyl)-1,2,4-triazin-3-amine
N-cyclopropyl-1,3-dimethyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-(quinazolin-4-yloxy)ethan-1-one
5-(2-fluorophenyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-{1-ethyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-1-methylpiperidine
1-(4-fluorophenyl)-4-[1-(propan-2-yl)piperidine-4-carbonyl]-1,4-diazepane
N,N-diethyl-2-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-4-(thiophen-2-yl)phenoxy)acetamide
6-(1-cyclopentylpiperidine-3-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
N-cyclopropyl-3-(3-fluorophenyl)-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}benzamide
methyl 4-(6-methyl-5-{[2-(methylsulfanyl)acetamido]methyl}-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl)benzoate
(2S,4R)-4-(4-{[1-(3-chlorophenyl)-N-methylformamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
3-(2-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}-2-oxoethyl)-6-methoxy-2,3-dihydro-1H-indol-2-one
N-[(7-{[5-(2-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-2-(3-fluorophenyl)acetamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-[4-(trifluoromethyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1S,5R)-3-(5-acetyl-4-methylpyrimidin-2-yl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(2-chlorophenyl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]morpholine-2-carboxamide
2-{4-[(6-fluoroquinolin-2-yl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
2-(5-chloro-2-methoxyphenyl)-2-[methyl(oxan-4-ylmethyl)amino]acetic acid
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]propan-1-one
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(2-hydroxypropyl)acetamide
N-cyclohexyl-2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-N-methyl-6-[4-(methylsulfanyl)phenyl]pyridine-3-carboxamide
3-[(3S,4R)-1-benzyl-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-N-(3-ethoxypropyl)propanamide
3-[(3,4-dimethylphenyl)methyl]-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-benzyl-6-(cyclopropylmethoxy)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-1,4-diazepan-2-one
N-[2-(4-fluorophenyl)ethyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
(3aR,6aR)-2-[(benzylcarbamoyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-6-[3-(methylsulfanyl)phenyl]pyridine-2-carboxamide
N-[(3S,4R)-1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-cyclohexyl-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[3-(4-phenoxybenzoyl)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
5-[3-(morpholin-4-yl)piperidine-1-carbonyl]quinoxaline
5-phenyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,2-oxazole-4-carboxamide
4-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholine
(2-{2-[1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
3-(4-methylphenyl)-N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
N-{1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
4-hydroxy-N-[(1R)-2-hydroxy-1-phenylethyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-(3-fluorobenzoyl)-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4,4,4-trifluorobutan-1-one
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
N2,N2-dimethyl-N4-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine