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7-(5-chloro-2-methoxyphenyl)-4-(furan-2-carbonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 5-{[1-(4-fluorophenyl)propan-2-yl]amino}-3-(2-methoxyacetamido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
7-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-N-(1,2-oxazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-cyclopropyl-1-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-(dimethylamino)-N-[(2-ethoxypyridin-3-yl)methyl]-4-methylpyrimidine-5-carboxamide
2-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyrimidine
(2S)-2-amino-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-phenylpropanamide
(1R,2S)-1-{2-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-imidazol-1-yl}-2,3-dihydro-1H-inden-2-ol
2-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
1-(2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)cyclopentanecarboxamide
5-butyl-4-(2-methoxypyridine-3-carbonyl)-1-(3-methylphenyl)piperazin-2-one
methyl (2S,4S)-4-(furan-2-amido)-1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidine-2-carboxylate
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[(1r,4r)-4-hydroxycyclohexyl]-1,2-oxazole-3-carboxamide
N-({1-[(3,5-dimethyl-1H-indol-2-yl)methyl]piperidin-3-yl}methyl)methanesulfonamide
N-methyl-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-(thiophen-3-ylmethyl)acetamide
N-[2-phenyl-2-(piperidin-1-yl)ethyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-(5-{[4-(diphenylmethyl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
2-{methyl[(4-methylphenyl)methyl]amino}-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]acetamide
2-(4-methylphenyl)-2-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}acetic acid
2-chloro-5-acetamido-N-[2-(1H-imidazol-4-yl)ethyl]benzamide
7-methyl-3-(piperidin-3-yl)-3,4-dihydroquinazolin-4-one
N-(furan-2-ylmethyl)-2-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]acetamide
5-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-N-(propan-2-yl)pyrimidin-2-amine
1-(oxan-4-yl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
3-({[2-(4-chlorophenoxy)ethyl](ethyl)amino}methyl)piperidin-3-ol
2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,3-dimethylfuran-2-carboxamide
1-(2-methoxy-5-{[(thiophen-3-ylmethyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
3-(3-methoxyphenyl)-N-{2-[methyl(phenyl)amino]ethyl}-1H-pyrazole-4-carboxamide
3-[(2,3-dimethoxyphenyl)methyl]-5-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
N,N-dimethyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
N-(1-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylfuran-2-carboxamide
2-(3-hydroxyazetidine-1-carbonyl)-6-(4-methoxyphenyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-(cyclopropylmethyl)-5-[2-(3-methoxyphenyl)acetyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4-(piperidin-3-ylmethyl)benzamide
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-(propan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
{[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(4-methoxyphenyl)methyl]methylamine
N3-ethyl-N5-(2-methylpropyl)-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(3-hydroxy-2,2-dimethylpropyl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[(5-methylthiophen-2-yl)methyl]propanamide
1-[1-(pyridin-2-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pent-4-en-1-one
5-(2-methoxyacetamido)-N-[(1R)-1-(4-methoxyphenyl)ethyl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
2-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-1H-1,3-benzodiazole
N-(6-cyanopyridin-3-yl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carboxamide
7-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 1-{9-methoxy-3-[(5-methylthiophen-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
N-{1-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
N,N-dimethyl-4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperazine-1-sulfonamide
N-[(2-chlorophenyl)methyl]-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(propan-2-yl)propanamide