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7-(2-methoxypyridin-3-yl)-1,2-dihydroisoquinolin-1-one
N-[(3,4-dimethoxyphenyl)methyl]-N-methyl-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
N5-[(2-methoxyphenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-ethyl-4-{3-[2-(3-fluorophenyl)ethyl]piperidine-1-carbonyl}piperidine
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amine
1-{5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
N-[3-(1H-indol-2-yl)phenyl]-1-(2-methylpropyl)piperidine-4-carboxamide
4-{4-[1-(4-chlorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}-1,4-oxazepane
4-[1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperidin-3-yl]benzoic acid
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-2-(methylamino)acetamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-ethyl-N-methylpiperidine-3-carboxamide
5-(1-benzoxepine-4-carbonyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidine-1-carbonyl}-6-phenyl-1,2-dihydropyridin-2-one
{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}[(4-fluorophenyl)methyl]amine
2-(4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}morpholin-2-yl)ethan-1-amine
2-(2-methoxyethyl)-9-{spiro[2.3]hexane-1-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
3-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-1-methyl-5-phenyl-1H-pyrazole
3-methanesulfonamido-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
ethyl 1-(5,8-dimethoxy-3-{[(thiophen-2-ylmethyl)amino]methyl}quinolin-2-yl)piperidine-4-carboxylate
2-(3-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}({[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl})amine
4-[2-methyl-7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,4-oxazepane
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[(1R)-1-(4-methoxyphenyl)ethyl]propanamide
3-{1-[1-(4-chlorophenyl)piperidin-4-yl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(3-fluorophenyl)-4H-1,2,4-triazole
1-benzyl-8-(1-hydroxypropan-2-yl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-phenyl-N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]benzamide
N-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-2-yl}ethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
6-(5-acetylthiophene-2-carbonyl)-N-[2-(3-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[(3S,4R)-3-propyl-4-[3-(pyridin-2-yl)propanamido]pyrrolidin-1-yl]propanoic acid
(2E)-3-(4-methoxyphenyl)-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}prop-2-enamide
{1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-fluorobenzamide
4-hydroxy-N,2-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]pyrimidine-5-carboxamide
N-[3-(1H-indazol-1-yl)propyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
5-(3,3-diethylpyrrolidine-1-carbonyl)-1-[(2-methoxyphenyl)methyl]piperidin-2-one
(2S)-4-methyl-2-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]formamido}pentanamide
3-[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
N-cyclopentyl-2-(2,5-dioxoimidazolidin-4-yl)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)acetamide
N-(4-ethoxyphenyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carboxamide
1-{2-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]ethyl}-1H-1,2,4-triazole
5-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridin-3-amine
8-[(3-chloro-4-hydroxyphenyl)methyl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-ethoxy-5-methyl-N-[(4-methyl-1,4-oxazepan-6-yl)methyl]benzene-1-sulfonamide
dimethyl[2-({[3-(pyrimidin-2-yloxy)phenyl]methyl}(thiophen-3-ylmethyl)amino)ethyl]amine
3-[(4-{furo[3,2-c]pyridin-4-yl}piperazin-1-yl)methyl]-7-methyl-1H-indole