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1-methoxy-8-(5-phenoxyfuran-2-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
{[(1R,5S,6S)-3-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
(3S,4R)-3-cyclopropyl-N,N-dimethyl-4-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamido]pyrrolidine-1-carboxamide
4-{[4-(cyclopentyloxy)phenyl]methyl}-N,N-dimethylpiperazine-1-sulfonamide
4-methyl-N-[3-(sulfamoylmethyl)phenyl]-1,4-diazepane-1-carboxamide
1-(2-{[(2,4-dimethoxyphenyl)methyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
3-(2,5-difluorobenzoyl)-1-(oxane-4-carbonyl)piperidine
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(pyrrolidin-1-yl)butan-1-one
1-[2-({[2-(furan-2-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
2-[(3S,4R)-3-methanesulfonamido-4-propylpyrrolidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
(1R,2S)-N1-propyl-N2-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}cyclohexane-1,2-dicarboxamide
1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carboxylic acid
2-(1-ethylpiperidin-4-yl)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
1-(4-methylquinazolin-2-yl)-N-[1-(thiophen-3-yl)propan-2-yl]piperidine-4-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-N,5-dimethyl-N-(1,2-oxazol-3-ylmethyl)-1H-pyrazole-4-carboxamide
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
(4-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}morpholin-3-yl)methanol
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-amine
3-fluoro-5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]benzonitrile
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-(naphthalen-2-ylmethyl)piperidin-3-ol
3-[(3R)-4-hydroxy-3-methylbutyl]-1-[2-(4-methoxyphenyl)phenyl]urea
N-[(5-methylfuran-2-yl)methyl]-1-oxo-2-[2-(pyridin-4-yl)ethyl]-2,3-dihydro-1H-isoindole-5-carboxamide
methyl 3-(5-chloro-2-fluorobenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2-{7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-2,3-dimethyl-N-(pyridin-2-ylmethyl)-1H-indole-5-carboxamide
(4aS,7aR)-1-[(4-methoxy-2-methylphenyl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-methyl-1'-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2S,4S)-1-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carboxamide
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-[methyl(piperidin-4-yl)amino]acetamide
2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]acetamide
N-[(5-ethylpyridin-2-yl)methyl]-N,5-dimethyl-2-(2-methylpropanamido)benzamide
5-ethyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrimidin-2-amine
5-[(isoquinolin-5-yloxy)methyl]-N-[(2R)-oxolan-2-ylmethyl]-1,2-oxazole-3-carboxamide
2-({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(ethyl)amino)ethan-1-ol
N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
ethyl 5-({[(3-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-4-methoxyphenyl)methyl]amino}methyl)furan-2-carboxylate
2-[3-(2-chlorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methylacetamide
methyl 3-{[(2,3-dimethoxyphenyl)formamido]methyl}-5-[(2E)-3-(3-fluorophenyl)prop-2-enamido]benzoate
2-[2-(4-chlorophenyl)morpholin-4-yl]-2-oxo-N-(propan-2-yl)acetamide
1-cyclohexyl-4-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
(1S,5R)-6-(pyridin-2-ylmethyl)-3-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2R,3R)-2-methoxy-1'-[(4-methoxy-2,3-dimethylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
5-(2-chlorophenyl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]furan-2-carboxamide
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-(oxan-2-ylmethoxy)acetamide
N-[(4-methylphenyl)methyl]-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
N-[3-(pyridin-3-yloxy)propyl]-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
N-(1-hydroxy-3-methylbutan-2-yl)-3,6,7-trimethyl-1-benzofuran-2-carboxamide
(3aR,5S,6S,7aS)-5,6-dihydroxy-N-[3-(trifluoromethyl)phenyl]-octahydro-1H-isoindole-2-carboxamide