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4-(4-cyclohexyl-1,4-diazepan-1-yl)-6-methoxypyrimidin-2-amine
3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
(1R,3S,5S)-8-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
7-(2-hydroxyethyl)-2-(5,6,7,8-tetrahydroquinoline-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-{1-[(2-ethoxyphenyl)methyl]-4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
2,6-dimethoxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
2-(methoxymethyl)-N,6-dimethyl-1-(naphthalen-1-ylmethyl)-4-oxo-N-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-[1-(1-{2-[3-(trifluoromethyl)phenyl]acetyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
N-benzyl-2-{2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
2-(4-methyl-1,4-diazepan-1-yl)-2-{4-[(morpholine-4-carbonyl)amino]phenyl}acetic acid
9-(5-ethyl-1,3-oxazole-4-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(6-methoxypyridin-3-yl)-4-methyl-1,2-dihydroquinolin-2-one
6-methyl-5-{2-oxo-2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[2-(4-acetylphenoxy)acetyl]-1-cyclohexyl-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-[(3,5-dimethylphenyl)methyl]-4-(4-fluoro-2-methylbenzoyl)piperazin-2-one
1-cyclohexyl-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
1-(diphenylmethyl)-4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
1-(furan-3-carbonyl)-4-[(5-methylthiophen-2-yl)methyl]-1,4-diazepane-6-carboxylic acid
1-(4-chlorobenzoyl)-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
[(2S,6S)-4-(2-chloro-6-fluoro-3-methylbenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
N-[(4-fluorophenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(2R,3R)-1'-[(2,4-dimethoxy-3-methylphenyl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1-(propan-2-yl)piperidine-4-carboxamide
N-{3-[methyl(phenyl)amino]propyl}oxane-2-carboxamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1H-pyrrole-2-carboxamide
4-(1-ethyl-1H-pyrazole-4-carbonyl)-1-(4-methoxyphenyl)-6,6-dimethylpiperazin-2-one
1-(cyclopropylmethyl)-6-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-{5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}phenol
3-methanesulfonamido-N-[(2-phenoxypyridin-3-yl)methyl]propanamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(5-methoxyfuran-2-carbonyl)piperidine-2-carboxamide
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(1H-imidazol-1-yl)ethan-1-one
2-methyl-N-[(5-methylpyrazin-2-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyrimidin-2-amine
5-(3-chloro-2-fluorobenzoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
(1R,3S)-7-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-7-azaspiro[3.5]nonane-1,3-diol
6-[methyl(pyrazin-2-ylmethyl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N,N-dimethyl-1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]azepan-4-amine
N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)cyclohexanecarboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
2-(2-oxopiperidin-1-yl)-N-[(3R,4S)-4-propyl-1-(pyridin-4-yl)pyrrolidin-3-yl]acetamide
N-({5-[(4-methoxy-2,5-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
[(2S)-1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
3-(cyclopropylmethyl)-5-[1-(2,3-dimethylbenzoyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
N-({7-[2-(2-chlorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
N-(1-benzoylpiperidin-4-yl)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carboxamide
5-ethyl-N4-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}pyrimidine-2,4-diamine
(2S)-2-acetamido-4-(methylsulfanyl)-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)butanamide
(3aS,6aS)-2-[(5-chlorofuran-2-yl)methyl]-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid