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8-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-cyclopropyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
5-methanesulfonyl-4-(piperidin-3-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]pyrimidin-2-amine
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-(hydroxymethyl)piperidin-1-yl]propan-1-one
1-{2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-2-oxoethyl}pyrrolidin-2-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[2-(4-fluorophenyl)piperidin-1-yl]propan-1-one
2-[9-(3-methoxybenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
3-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-3,9-diazaspiro[5.5]undecane
2-hydroxy-N-[(3R,4S)-4-phenyl-1-(3,3,3-trifluoropropyl)pyrrolidin-3-yl]acetamide
N-benzyl[(3,5-dimethoxyphenyl)amino]sulfonamide
2-fluoro-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}-5-sulfamoylbenzamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
2-(cyclopent-2-en-1-yl)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
1-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]-6-methylpyridine-3-carboxylic acid
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(3,4-dichlorophenyl)ethan-1-one
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
3-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
6-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methyl-N-(2-methylpropyl)acetamide
2-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
1-(cyclohexylmethyl)-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
3-{4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazin-1-yl}benzoic acid
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(2-fluorophenoxymethyl)piperidine
2-methoxy-N-methyl-5-({[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]carbamoyl}amino)benzamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
methyl 1-ethoxy-2-oxo-8-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
1-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]ethan-1-one
ethyl 1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-[(5-ethylpyridin-2-yl)methyl]-1-methylurea
1-[1'-(3-chlorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-(2-ethoxyphenyl)-N'-methyl-N'-[2-(oxan-4-yl)ethyl]propanediamide
6-methyl-2-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
methyl 2-{1-[1-ethyl-5-(2-methoxyacetamido)-2-(pyridin-3-yl)-1H-1,3-benzodiazol-7-yl]-N-methylformamido}acetate
4-{1-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-imidazol-2-yl}pyridine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(2-chlorophenoxy)ethan-1-one
2-ethyl-8-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
(2R,3S,6R)-3-phenyl-5-(pyridin-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4-methoxyphenyl)-4-[4-(2-methylpropyl)benzoyl]piperazin-2-one
N-(2-{3-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]phenoxy}propyl)imidazo[1,2-a]pyridine-2-carboxamide
9-[(2R)-2-hydroxy-3-methylbutanoyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(2,5-dioxoimidazolidin-1-yl)-N-methylacetamide
N-({3,5-dimethoxy-4-[2-(1-methylpyrrolidin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzenesulfonamide
1-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]piperidine-4-carbonitrile
N2,N2-dimethyl-N4-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
1-({5-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
1-[4-(3-methoxyphenyl)phenyl]-N-(1-methyl-1H-pyrazol-5-yl)piperidin-4-amine
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(2-methylbenzamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
N-({8-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)cyclohexanecarboxamide