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(4aS,8aR)-6-(pyrazin-2-yl)-1-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-amino-N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-4-methylpyrimidine-5-carboxamide
methyl 2-({[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)amino)acetate
4-hydroxy-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-2-(thiophen-2-yl)pyrimidine-5-carboxamide
3-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-3-(2-methylphenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
2-methyl-5-{[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]sulfanyl}-1,3,4-thiadiazole
6-chloro-N,N-dimethyl-3-[({2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}amino)methyl]imidazo[1,2-a]pyridine-2-carboxamide
2-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
2-(pyridin-3-yl)-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]pyrimidine
1-[3-(oxolan-3-yl)propyl]-4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazole
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-cyclopropyl-3-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]propanamide
N-[2-(3-methoxyphenyl)phenyl]-1-(pentan-3-yl)piperidine-4-carboxamide
N-[(2R,3R)-2-methoxy-1'-[3-(5-methylfuran-2-yl)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-hydroxyethan-1-one
5-oxo-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
8-methoxy-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-tert-butyl-6-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)phenol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]acetamide
({5-[1-(4-cyclopentylpyrimidin-2-yl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
1-(2-methoxyphenyl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-pyrazole-4-carboxamide
methyl 3-[(3,4-dimethylphenyl)methyl]-7-oxo-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-chloro-4-{[1-(cyclopropylmethyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
4-{1-[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}morpholine
4-{1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}quinoline
2-(3-fluorophenoxymethyl)-N-[(3-methyl-1-benzofuran-2-yl)methyl]-1,3-oxazole-4-carboxamide
methyl[1-(pyridin-4-yl)ethyl]{[2-(trifluoromethoxy)phenyl]methyl}amine
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-(1,3-benzothiazol-2-ylmethyl)-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-cyclopentyl-N-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
9-(cyclopropylmethyl)-4-[4-(dimethylamino)pyrimidin-2-yl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
7-(3,6-dimethylpyrazin-2-yl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(2,4-dioxoimidazolidin-1-yl)-N-[(2-methylphenyl)(pyridin-4-yl)methyl]benzamide
(2S,4R)-N-ethyl-4-[2-(methylsulfanyl)acetamido]-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl][(3,5-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
{5-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl}(phenyl)methanol
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2,2-dimethylpropan-1-one
6-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
3-[1-(furan-2-ylmethyl)piperidin-4-yl]-1-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methyl-2-(1H-pyrrol-1-yl)propanamide
3-(diphenylmethyl)-N-(1H-imidazol-2-ylmethyl)-N-methyl-1,2-oxazole-5-carboxamide
methyl 3-(2,5-dimethylbenzoyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-(pyridin-3-yl)pyrimidin-2-amine
6-[4-(1H-pyrazol-3-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-(2-hydroxybutyl)-2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-{5-[2-(2-hydroxyethyl)piperidine-1-carbonyl]-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazol-7-yl}cyclobutanecarboxamide
N-cyclopropyl-1-[(1s,4s)-4-[2-(2-chloro-4-fluorophenyl)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-hydroxy-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)benzamide