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N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-hydroxy-2-(3-methylphenyl)pyrimidine-5-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-(4-hydroxyphenyl)-5-oxopyrrolidine-3-carboxamide
methyl({[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
1-{1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]piperidin-4-yl}piperidin-4-ol
N-{3-[methyl(phenyl)amino]propyl}-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(2-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
2-[2-(pyridin-3-yl)ethyl]-9-(thiophene-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[3,3-dimethyl-1-(pyridin-3-yl)butyl]amino}-N-(2,4-dimethylphenyl)acetamide
(1S,5R)-6-(cyclopropylmethyl)-3-(3-fluoro-4-methylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
4-methyl-2-{2-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
4-ethyl-5-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-thiazol-2-amine
N,4-dimethyl-3-[({[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}carbamoyl)amino]benzamide
2-(dimethyl-1,2-oxazol-4-yl)-1-{4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
4-{2-[3-(dimethylamino)pyrrolidin-1-yl]acetyl}-1-(3-methoxyphenyl)piperazin-2-one
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}phenol
1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-(methylamino)ethan-1-one
3-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
1,3-dimethyl-N-[3-(oxolan-3-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-1-(2-methylpiperidin-1-yl)propan-1-one
1-[3-(2-chlorophenyl)pyrrolidin-1-yl]-2-(furan-2-yl)ethane-1,2-dione
3-(azepane-1-carbonyl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(2H-1,3-benzodioxol-5-yl)-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-3-amine
5-chloro-2-methyl-6-[3-(2-methylpropoxy)phenyl]pyrimidin-4-ol
1-{1-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,3-benzodiazole
3-[(dimethylamino)methyl]-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-3-ol
(3S,4S)-4-methyl-1-(quinolin-4-yl)piperidine-3,4-diol
1-methyl-6-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-[(2-methoxyphenyl)methyl]-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
5-amino-3-(1-phenyl-1H-pyrazol-5-yl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-{[4-(butan-2-yloxy)-3-chloro-5-methoxyphenyl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
(3S)-3-({5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)azepan-2-one
4-{[1-(3-phenylpropyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
N-[1-(4-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]cyclopentanecarboxamide
3-benzyl-8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
2-cyclobutyl-N-[(2,5-dimethoxyphenyl)methyl]-5-(2-methoxyacetamido)-1-methyl-1H-1,3-benzodiazole-7-carboxamide
2-phenyl-N-{[8-(pyridin-3-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
[(2-chloro-5-ethoxy-4-propoxyphenyl)methyl][1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]amine
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(thiophen-2-yl)ethan-1-one
3,5-dimethoxy-N-{[1-(pent-4-enoyl)piperidin-3-yl]methyl}benzamide
methyl 5-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-[6-(benzyloxy)pyridin-3-yl]-5-(methanesulfonylmethyl)pyridine
2-ethyl-N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}pyrimidine-5-carboxamide
3-(4-acetyl-6-hydroxy-1,4-diazepane-1-carbonyl)-1,2-dihydroquinolin-2-one
methyl 3-{[2-(1H-indol-3-yl)acetamido]methyl}-5-(2-methoxybenzamido)benzoate
1-{5-[(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}butan-2-ol
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide