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N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-3-(1H-pyrazol-1-yl)benzamide
8-[(2S)-2-hydroxypropanoyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-(4-benzylpiperazine-1-carbonyl)-6-[(5-ethylfuran-2-yl)methyl]-6-azaspiro[2.5]octane
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-(4,6-dimethylquinazolin-2-yl)piperidine-4-carboxamide
6-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]pyridine-2-carbonitrile
2-[(4-benzylpiperazin-1-yl)methyl]-N-methyl-N-(1H-pyrazol-5-ylmethyl)-1,3-oxazole-4-carboxamide
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-1-[(2-methoxyphenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
2-(2-methoxyethyl)-1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
3-benzoyl-1-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
N-[1-ethyl-2-(2-fluorophenyl)-5-(4-propylpiperazine-1-carbonyl)-1H-1,3-benzodiazol-7-yl]acetamide
4-benzyl-3-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-2,6,8-trimethylquinoline
2-(dimethyl-1,2-oxazol-4-yl)-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}acetamide
5-ethyl-5-{1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl}-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
1-(4-methoxybenzenesulfonyl)-N-(pyrimidin-2-yl)azepan-3-amine
(1R,5R)-6-[2-(benzenesulfonyl)ethyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]azepan-4-amine
methyl 3-{[1-(1-methylpiperidin-4-yl)piperidin-3-yl]carbamoyl}benzoate
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
3-(dimethyl-1,2-oxazol-4-yl)-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
ethyl 1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
N-[4-(azepan-1-yl)butyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-(3-propoxypiperidin-1-yl)pyrimidine
N-methyl-N-{3-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-oxopropyl}methanesulfonamide
3-(4-methoxyphenyl)-N-methyl-3-phenyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
4-(4-{1-[N-methyl-2-(1H-pyrazol-1-yl)acetamido]-2-(2-methylphenyl)ethyl}piperidine-1-carbonyl)pyridin-1-ium-1-olate
butyl 7-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
3-(azepane-1-carbonyl)-N-(2,3-dihydro-1H-inden-2-yl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[1-benzyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-1,5,5-trimethylpyrrolidin-2-one
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-5,6-dimethylpyrimidin-4-amine
3-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperidin-3-yl}benzoic acid
7-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-oxo-1H,2H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
3-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-4-methyl-1,2,5-oxadiazole
1-{3-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{4-[(3,5-difluorophenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
8-[(3,4-dimethylphenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
1-[3-(methylsulfamoyl)phenyl]-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
methyl 3-(2,1,3-benzothiadiazol-5-ylmethyl)-9-(benzyloxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-methoxy-N-{2-[3-(1H-pyrazol-3-yl)phenyl]phenyl}acetamide
N-(1-methanesulfonylpiperidin-4-yl)-3-(piperidin-4-ylmethyl)benzamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
ethyl 1-(cyclopent-1-ene-1-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylate
2,2-dimethyl-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}thiomorpholin-3-one
1-(1,2,3-thiadiazole-4-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N,1-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrrole-2-carboxamide
3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydroquinolin-2-one
1-phenyl-5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1H-1,2,3,4-tetrazole
N-(2-hydroxyethyl)-3-(5-methylfuran-2-yl)-N-(1,3-thiazol-2-ylmethyl)benzamide
(1S,5R)-6-benzyl-3-[2-(methylsulfanyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]but-3-en-1-one