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(3S,4R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
5-(2-{4-[(3,4-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-tert-butyl-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
9-(1H-1,3-benzodiazol-2-ylmethyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
1-(azocan-1-yl)-3-[5-({[(1-ethyl-1H-imidazol-2-yl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
(2S)-2-amino-N-[(2-methoxyphenyl)methyl]-4-(methylsulfanyl)-N-propylbutanamide
3-{1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]piperidin-3-yl}benzoic acid
1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
8-(furan-3-ylmethyl)-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(cyclopropylmethyl)-1-[2-(methylamino)pyridine-3-carbonyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-cycloheptyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-[(2-chlorophenyl)methyl]-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
methyl 6-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}pyrimidine-4-carboxylate
N-(3,4-difluorophenyl)-6-[(5-acetamidothiophen-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
ethyl 6-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylate
1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(3-methylphenoxy)piperidine
6-methyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[3-(4-fluorophenoxy)piperidin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{2-[2-(trifluoromethyl)phenyl]ethyl}propanamide
8-[(2,3-difluorophenyl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}pyrrolidin-3-yl)acetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-(pyrrolidine-1-sulfonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,1,3-trimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-ethyl-N-[2-(3-fluorophenyl)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
N-[(2-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)cyclobutanecarboxamide
4-(4-methoxyphenyl)-3-(2-phenylethyl)-4H-1,2,4-triazole
3-[(4aR,7aS)-4-[methyl(phenyl)carbamoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
(1R,5S,6R)-3-({3-[(4-ethylpiperazin-1-yl)methyl]-2,5-dimethylphenyl}methyl)-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
1-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}piperidine-3-carbonitrile
1-(cyclopropylmethyl)-3-({[(dimethyl-1,3-thiazol-2-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
2-[2-(4-benzyl-6-methoxy-3-oxo-1,4-diazepan-1-yl)-2-oxoethyl]-4-phenyl-1,2-dihydrophthalazin-1-one
N-({7-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)methanesulfonamide
4-{6-[1-(4-ethyl-5-methylpyrimidin-2-yl)piperidin-3-yl]-2-methylpyrimidin-4-yl}morpholine
(4aR,7aS)-1-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-4-(thiophene-2-sulfonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl (2S)-2-(3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamido)-2-phenylacetate
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazole-5-carboxamide
N,N-dimethyl-4-[2-(naphthalen-1-ylmethyl)morpholine-4-carbonyl]piperidine-1-carboxamide
2-methyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{2-[3-(3-methoxypropyl)piperidin-1-yl]pyridine-4-carbonyl}-4-methylpiperazine
2-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)ethan-1-one
5-oxo-1-(pyridin-4-ylmethyl)-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)pyrrolidine-3-carboxamide
{9-[(2-aminopyridin-3-yl)methyl]-3-cyclopentanecarbonyl-3,9-diazaspiro[5.5]undecan-1-yl}methanol
1-(3-phenylpropyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-3-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one