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2-(3,5-difluorophenyl)-1-(4-{5-[(1E)-prop-1-en-1-yl]-2-(pyridin-3-yl)pyrimidin-4-yl}piperidin-1-yl)ethan-1-one
N-[2-ethyl-4-(4-methanesulfonylphenyl)phenyl]acetamide
3-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-(4-ethoxy-2-fluorophenyl)urea
2-{4-[(4-methoxynaphthalen-1-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
3-(1-{1-[(3-chloro-2-fluorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-1-ol
2-methyl-N-{[3-(3-methylpyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}aniline
2-methyl-8-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-[2-(N-methylmethanesulfonamido)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-({3-methyl-7-[4-(1H-pyrazol-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
3-{5-[(2E)-but-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
4-[4-(pyrrolidine-1-carbonyl)phenoxy]-1-(1,3-thiazol-2-ylmethyl)piperidine
(2S,4S)-N,N-diethyl-4-[(3E)-pent-3-enamido]-1-(pyridine-4-carbonyl)pyrrolidine-2-carboxamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-(piperidin-1-yl)butanamide
8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-1-(2-phenylethyl)piperidine
2-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-(6-aminohexyl)-[1,2,4]triazolo[4,3-a]pyridine-7-carboxamide
3-butanamido-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidine
2-[2-(dimethylamino)ethyl]-8-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)[(5-methylfuran-2-yl)methyl]amine
3-(4-{2-[4-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidine-1-carbonyl)pyridine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]acetamide
N-(2,2-dimethyloxan-4-yl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
2-(methylsulfanyl)-4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
(2S)-2-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}amino)propanamide
N,N-dimethyl-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-sulfonamide
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-(furan-2-ylmethyl)pyrrolidin-2-one
1-{2-hydroxy-5-[2-(morpholin-4-ylmethyl)phenyl]phenyl}ethan-1-one
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
3-[(1H-1,3-benzodiazol-2-ylmethyl)amino]-N-(pyridin-2-ylmethyl)-5-(pyrrolidine-1-sulfonyl)benzamide
5-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)imidazolidine-2,4-dione
8-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(2-hydroxyethyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1H-1,3-benzodiazole-5-carboxamide
3-benzyl-4-(2,3-difluoro-4-methylbenzoyl)piperazin-2-one
6-[(3-methylpyridin-4-yl)methyl]-5,6-dihydro-1,6-naphthyridin-5-one
2-methoxy-6-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
2-(dimethylamino)-8-(1,3-thiazol-4-ylmethyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-(cyclopropylmethyl)-2-oxo-3-{1-[(pyridin-2-yl)carbamoyl]ethyl}-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
N-cyclopropyl-N-{[3-(oxan-2-ylmethoxy)phenyl]methyl}quinoline-2-carboxamide
4-(2-chlorophenoxy)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
[1-(2-fluorophenyl)propan-2-yl]({[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl})amine
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[(2,3-difluoro-4-methylphenyl)methyl]propanamide
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
methyl (1R,3S,3aR,6aS)-3-(3-fluoropyridin-4-yl)-5-methyl-1-(2-methylpropyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-[5-({[(2-chlorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
3-[1-(2-methoxyacetyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
8-(1-benzofuran-2-ylmethyl)-3-[2-(dimethylamino)ethyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione