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N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-2-(2-chloro-4-fluorophenyl)acetamide
8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(1H-1,3-benzodiazol-1-yl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)methanol
methyl 4-({[6-oxo-1-(pyridin-2-ylmethyl)piperidin-3-yl]formamido}methyl)benzoate
1-(5-acetylthiophene-2-carbonyl)-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
3-(but-2-yn-1-yl)-5-{1-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
(4aS,7aR)-1-[2-(1,2-benzoxazol-3-yl)acetyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-(2-hydroxybutyl)-6-(4-methoxyphenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-5-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
2-(4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}morpholin-3-yl)acetic acid
4-{[(2-cyclohexylpyrimidin-5-yl)methyl]amino}-1-phenylpyrrolidin-2-one
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
2-[3-cyclopentyl-5-(6-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(2-methylphenyl)sulfanyl]piperidine
1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
N-[(5-chloro-1H-indol-2-yl)methyl]-1-cyclopropyl-6-oxopiperidine-3-carboxamide
3-(2-methylphenyl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
N-[4-(pyridin-2-yl)butyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
(1S,6R)-9-(3-methoxybenzenesulfonyl)-3,9-diazabicyclo[4.2.1]nonane
3-[2-(benzyloxy)ethyl]-9-(furan-2-carbonyl)-3,9-diazaspiro[5.5]undecane
N-cyclopropyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)oxolane-2-carboxamide
6-{3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-4-(1H-1,2,4-triazol-3-yl)benzamide
7-[4-(benzyloxy)butanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(2-{[4-(thiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrrol-1-yl)pyridine
ethyl 4-{6,7-dimethoxy-3-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]quinolin-2-yl}piperazine-1-carboxylate
3-{1-[3-(1H-imidazol-4-yl)propanoyl]piperidin-4-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
2-(methylamino)-N-[2-(3-phenylpiperidin-1-yl)ethyl]pyridine-4-carboxamide
{[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
3,7-dimethyl-11-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,7,11-triazaspiro[5.6]dodecane
N-[(2-fluorophenyl)methyl]-3-{1-[3-(2-oxopyrrolidin-1-yl)benzoyl]piperidin-3-yl}propanamide
1-methyl-4-({4-[3-methyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenyl}methyl)piperazine
6-(2-chlorobenzoyl)-N-[2-(3-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
8-(2H-1,3-benzodioxol-5-ylmethyl)-1-(2-methoxyethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyrimidine-2-carboxamide
2-{5-[(1,1-dioxo-1λ6-thian-4-yl)methyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}acetic acid
1-{3-[3-(2-fluorophenoxy)azetidine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(5-methylpyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-N-(2,3-dimethylphenyl)acetamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]propan-1-one
9-methoxy-7-oxo-3-(2,2,3,3-tetramethylcyclopropanecarbonyl)-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(3-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}phenyl)-4-phenylbutanamide
N-(1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-methyl-1-oxopropan-2-yl)thiophene-2-carboxamide
4-(1-butyl-1H-1,2,4-triazol-5-yl)-1-ethyl-1,2-dihydropyridin-2-one
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-5-(1H-1,3-benzodiazol-1-ylmethyl)-1H-pyrazole-3-carboxamide
N-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
5-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid