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2-acetamido-3-methyl-N-({5-methyl-2-[3-(3-methylbutanamido)phenyl]-1,3-oxazol-4-yl}methyl)butanamide
2,3,6-trimethyl-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]quinoline-4-carboxamide
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}[(5-ethylpyridin-2-yl)methyl]methylamine
3-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
(2R,3R)-3-({2-[cyclopentyl(methyl)amino]ethyl}(methyl)amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-({1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
N-[3-(4-{[2-(dimethyl-1,2-oxazol-4-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-2-(4-methylphenoxy)acetamide
3-(azepane-1-sulfonyl)-5-(2,4-dimethyl-1H-imidazol-1-yl)benzoic acid
2-[4-(4-methylpent-3-en-1-yl)-1-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
5-(2-methylpropyl)-1'-(thiophen-3-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-N-(furan-2-ylmethyl)acetamide
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-2-phenoxyacetamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-[4-(methylsulfanyl)phenyl]acetamide
N,N-dimethyl-3-oxo-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decane-8-sulfonamide
1-acetyl-4'-(3,3-dimethylbutyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[2-(3-fluorophenyl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidin-2-one
2-cyclobutyl-N-[(5-fluoro-2-methylphenyl)methyl]-1-methyl-7-(oxolane-2-amido)-1H-1,3-benzodiazole-5-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}propanamide
N-(butan-2-yl)-N-{[1-(pyrimidin-2-ylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}acetamide
3-(5-{[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}thiophen-2-yl)prop-2-yn-1-ol
7-fluoro-3-methyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-benzofuran-2-carboxamide
1-{4-[(4-ethylpyridin-2-yl)amino]piperidin-1-yl}ethan-1-one
6-(1-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}piperidin-3-yl)-2-methylpyrimidin-4-ol
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-(thiophen-2-ylmethyl)-4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-1,4-diazepane
methyl (2S,4R)-1-[(4-fluorophenyl)methyl]-4-(quinoline-2-amido)pyrrolidine-2-carboxylate
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(2,5-dimethoxyphenyl)acetamide
9-(1H-imidazole-2-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(dimethylamino)-2-(2-fluorophenyl)-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
ethyl 4-[ethyl({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})carbamoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepan-5-one
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2,6-dimethylquinoline-4-carboxamide
3-[2-(ethanesulfonyl)ethyl]-1-(3-ethylphenyl)urea
N-[(2,3-difluorophenyl)methyl]-4-methyl-5-(1-methyl-1H-pyrazol-3-yl)-1,3-thiazol-2-amine
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-[1-(pyridin-4-yl)propyl]-1,2-oxazole-3-carboxamide
{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
methyl 2-({[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}(cyclopropyl)sulfamoyl)benzoate
2-methylpropyl N-methyl-N-({1-[(3S,5S)-5-(methylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)carbamate
methyl 3-(2-chlorobenzamido)-5-{[(1-methyl-1H-pyrazol-5-yl)formamido]methyl}benzoate
N-[(2,4-dimethoxyphenyl)methyl]-3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
2-methyl-7-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(2-chlorophenyl)methyl]-N-(prop-2-en-1-yl)-1H-1,2,3-benzotriazole-5-carboxamide
N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-4-(3-fluorophenyl)benzamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]pent-4-enamide
4-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-6-methoxypyrimidin-2-amine
2-chloro-N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}pyridine-4-carboxamide
N-methyl-N-(quinoxalin-6-ylmethyl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-cyclohexyl-4-[2-(3-methyl-1H-1,2,4-triazol-5-yl)acetyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one