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3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}propanamide
3-(1H-indol-3-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-methoxyethan-1-one
4-(4-chlorobenzoyl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(4-chlorophenyl)ethyl]-1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carboxamide
2-(2-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}phenoxy)-1-(4-methylpiperidin-1-yl)ethan-1-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cyclohexyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxamide
7-[(2-chloro-6-fluorophenyl)methyl]-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-benzyl{[5-methoxy-2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]amino}sulfonamide
2-(4-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)pyrazine
3-({[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-{1-[4-(dimethylamino)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
4-[1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)piperidin-3-yl]benzoic acid
(1S,5R)-6-(cyclopropylmethyl)-3-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(furan-3-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
5-{[3-(1H-1,3-benzodiazol-2-yl)azetidin-1-yl]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
N-[(2-aminopyrimidin-5-yl)methyl]-2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
4-(furan-3-ylmethyl)-3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
2-{4-cyclohexyl-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
methyl 1-(benzyloxy)-8-[(2-chloro-3,4-dimethoxyphenyl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-(pyridin-3-ylmethyl)benzene-1-sulfonamide
(4-{[1-(dimethyl-1,3-thiazole-5-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-(2,2,2-trifluoroethyl)-1,4-dihydropyridine-3-carboxamide
2-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
3-(2-methoxyethyl)-1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidine-3-carboxylic acid
2-benzyl-8-[2-(pyrrolidin-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
methyl 3-(3-chlorobenzoyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2,3-dimethyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]quinoxaline-6-carboxamide
2-[4-(4-acetylphenyl)piperazin-1-yl]-N,N-dimethyl-6-(4-methylthiophen-2-yl)pyridine-3-carboxamide
(4aS,8aR)-6-(dimethyl-1,3-oxazole-5-carbonyl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
6,7-dimethoxy-2-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
methyl[(2-methylpyridin-4-yl)methyl]{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
3-(2-phenylethyl)-5-(1H-pyrazol-4-yl)-1,2,4-oxadiazole
1-({2-[3-(1-hydroxyethyl)phenyl]phenyl}methyl)piperidin-4-one
1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(4-phenoxybenzoyl)piperidine
3-(4-chlorophenyl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-3-phenylpropanamide
3-(1H-1,3-benzodiazol-2-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-(3-fluoro-4-hydroxyphenyl)-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]acetamide
N-{3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}naphthalene-2-sulfonamide
1-cyclopropyl-5-oxo-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]pyrrolidine-3-carboxamide
N-[(2,3-difluorophenyl)methyl]-1-(4,6-dimethylquinazolin-2-yl)piperidin-4-amine
N-[4-({4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)phenyl]acetamide
4-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-2-methyl-6-(2-methylpropyl)pyrimidine
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine