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N-{[7-(2H-1,3-benzodioxole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}propane-1-sulfonamide
N-[(2R,3R)-1'-(2-cyclohexylacetyl)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-N,N-dimethyl-6-(4-methylthiophen-2-yl)pyridin-2-amine
1-(2-methoxyphenyl)-3-(propan-2-yl)-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methoxypiperidine
2-{[(3R,5S)-1-[(2-chlorophenyl)methyl]-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]sulfanyl}-4,6-dimethylpyrimidine
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(1-oxo-4-phenyl-1,2-dihydrophthalazin-2-yl)acetamide
5-{[1-(2-phenylethyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
4-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,4-diazepan-5-one
N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,5-dimethylbenzamide
(cyclobutylmethyl)({[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
N'-(3-fluorophenyl)-N-[(1-methylpyrrolidin-3-yl)methyl]butanediamide
4,6-dimethyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl (2S)-2-{[1-(4,6-dimethylquinazolin-2-yl)piperidin-4-yl]formamido}-3-methylbutanoate
N-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-4-(pyridin-4-yl)piperidine-1-carboxamide
1-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-3-(1,3-dihydro-2-benzofuran-5-yl)urea
5-chloro-6-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}pyridine-3-carboxylic acid
8-methyl-3-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-3,4-dihydroquinazolin-4-one
N-methyl-N-[2-(oxan-2-yl)ethyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
2,5-difluoro-N-(1-{7-[(3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
6-(2-methoxyphenyl)-N-[3-(propan-2-yloxy)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-{[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
N-{2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}-4-fluorobenzamide
N-methyl-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
N-[2-(4-methoxyphenyl)phenyl]-1-(2-phenylethyl)piperidine-3-carboxamide
3-methoxy-N-methyl-4-[(1-methylpiperidin-4-yl)oxy]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide
9-(cyclopropylmethyl)-1-methyl-4-[2-oxo-2-(piperidin-1-yl)ethyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-5-fluoropyridine
1-(3-methoxybenzoyl)-4-(oxane-4-carbonyl)piperazine
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]acetamide
2-[methyl(pyridin-4-ylmethyl)amino]-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}ethan-1-one
3-(2-methoxyphenyl)-1-(3-methoxypropyl)-3-{2-oxo-2-[2-(pyridin-3-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
N-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}methyl)-3-methylfuran-2-carboxamide
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-4-methylpentan-1-one
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-methyl-N-(2-phenoxyethyl)benzamide
4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-2-(trifluoromethyl)morpholine
8-fluoro-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]quinoline-2-carboxamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
6-{[ethyl(methyl)amino]methyl}-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1,2-dihydropyridine-3-carboxamide
1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
8-{[3-(methylsulfanyl)phenyl]methyl}-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
3-benzyl-N-(2,3-dihydro-1H-inden-1-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(2-methoxyethyl)-1-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(furan-2-ylmethyl)propanamide
1-[3-(azepane-1-carbonyl)phenyl]-3-ethyl-3-[(5-methylfuran-2-yl)methyl]urea
2-[1-methyl-4-(6-methylpyridazin-3-yl)-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
1-[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]pyrrolidin-2-one
4-phenyl-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]butan-1-one