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2-(pyridin-4-ylsulfanyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide
N-[2-(3-fluorophenyl)ethyl]-2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
4-[(1R)-1-(4-fluorophenyl)ethyl]-3-(1-methyl-1H-pyrazol-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(4-{[2-(3-chlorophenoxy)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]cyclobutanecarboxamide
5-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
N-[2-(3-chlorophenyl)ethyl]-5-(2-ethylpiperidine-1-carbonyl)-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(1-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)-N-cyclopropylpyridine-2-carboxamide
7-(cyclohex-1-en-1-yl)-4-{imidazo[1,2-a]pyridine-2-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{1-[1-(pyridin-4-yl)propyl]-1H-imidazol-2-yl}quinoline
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
3-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-N-(2,5-dimethoxyphenyl)-3-oxopropanamide
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}acetamide
N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-2,3-dimethylquinoxaline-6-carboxamide
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
methyl 5-(cyclobutylamino)-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4,4,4-trifluoro-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}butanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperidin-3-ol
5-[2-(1-carbamoylethoxy)phenyl]thiophene-2-carboxylic acid
N-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-7-oxo-3-(pent-4-enoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
2-[cyclopentyl(methyl)amino]-1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)ethan-1-one
{3-[(4-fluorophenyl)methyl]-1-(quinolin-2-yl)piperidin-3-yl}methanol
2-[2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
methyl 1-{[3-(furan-2-amido)-2-(methoxycarbonyl)thieno[2,3-b]pyridin-6-yl]methyl}piperidine-2-carboxylate
2-[(1S,5R)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
2-(2,3-dichlorophenyl)pyridine-4-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(2-methylfuran-3-carbonyl)piperidin-3-yl]piperazine
3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-[3-(2-oxopyrrolidin-1-yl)phenyl]urea
N-[(3-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-cyclopropyl-2-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]pyridine-4-carboxamide
3-(4-fluoro-3-methylphenyl)-1-methyl-6-(quinolin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[2-(1-{[(2,3-dimethylphenyl)carbamoyl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)ethyl]acetamide
5-methanesulfonyl-N,2-dimethyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidin-4-amine
4-(4-{3-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-ylmethyl]phenoxy}butyl)morpholine
5-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)-1,3-benzothiazol-2-amine
(2S)-1-[2-(adamantan-1-yl)acetyl]pyrrolidine-2-carboxylic acid
7-methoxy-2-[3-(4-methoxypiperidine-1-carbonyl)piperidin-1-yl]-4-methylquinazoline
5-acetamido-1-(2-methoxyethyl)-N-(3-methylbutyl)-2-(pyridin-2-yl)-1H-1,3-benzodiazole-7-carboxamide
3-(3-chloro-2-fluorophenyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]urea
3-cyclopropyl-4-(3,5-dimethyl-1-benzofuran-2-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3,5,7-trimethyl-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-1H-indole-2-carboxamide
[(3R,4R)-1-(2,3-dimethyl-1H-indole-7-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
4-amino-2-[3-(benzyloxy)phenyl]pyrimidine-5-carbonitrile
methyl 5-[(2,2-dimethylpropyl)amino]-3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3,4-dimethoxyphenyl)methyl]-7-acetamido-N-methyl-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
4-(dimethyl-1,3-oxazole-4-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
N-[(3R,4S)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]cyclobutanecarboxamide