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(5S,9aS,9bS)-5-(2-chloro-4,5-dimethoxyphenyl)-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(2,5-dimethoxyphenyl)-N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}acetamide
N-[(3-chlorophenyl)methyl]-2-(4-methylpiperazin-1-yl)-6-(thiophen-2-yl)pyridine-3-carboxamide
N-[2-(2-fluorophenyl)-1-[1-(3-methoxybenzoyl)piperidin-4-yl]ethyl]-N,2-dimethylfuran-3-carboxamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-methyl-N-(2-phenylethyl)piperidin-4-amine
2-cyclopentyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
8-[2-(dimethylamino)ethyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl 3-(1-methylcyclohexanecarbonyl)-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]acetamide
1-(2-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-(thiolan-3-yl)pyridin-2-amine
(2S,4R)-N-ethyl-1-[(2E)-2-methylbut-2-en-1-yl]-4-(2-oxo-2-phenylacetamido)pyrrolidine-2-carboxamide
methyl 1-(3-{4-[(2,2-dimethyl-3-oxopiperazin-1-yl)methyl]phenoxy}-2-hydroxypropyl)piperidine-4-carboxylate
2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
5-acetyl-N-[(4-sulfamoylphenyl)methyl]thiophene-3-carboxamide
3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]-1-(thiophen-3-ylmethyl)piperidine
{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
5-(1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1,7-dimethyl-1H-indole-2-carboxamide
3-(azetidine-1-sulfonyl)-N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]benzamide
(3S,7S)-5-[4-(dimethylamino)benzoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
4-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]benzonitrile
(3aR,6aR)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(2-methoxyacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
8-(2-ethoxyacetyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-methoxy-N-(2-methoxyethyl)-2-{[1-(2-phenylpropyl)piperidin-4-yl]oxy}benzamide
4-{2-methyl-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carbonyl}-1-(4-methylphenyl)piperazin-2-one
methyl 3-({[2-(2-cyclobutaneamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}carbamoyl)benzoate
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
5-{[(2-hydroxy-2-phenylethyl)(methyl)amino]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
4-(benzyloxy)-1-{3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidine
(2S)-N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
2-[(5-chloro-2,3-dimethoxyphenyl)methyl]-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
4-[2-(1-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]phenol
1-(1,3-oxazole-4-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-fluoro-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-5-sulfamoylbenzamide
N-{[5,8-dimethoxy-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2H-1,3-benzodioxole-5-carboxamide
1-benzyl-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-[4-(2-fluorophenyl)-1H-pyrazol-5-yl]-1-(furan-2-ylmethyl)piperidine
5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(2-methylbutyl)piperidin-4-yl]imidazolidine-2,4-dione
1-[(2-methoxyphenyl)methyl]-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
6-methyl-2-{1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carbonitrile
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[1-(thiophen-3-yl)propan-2-yl]piperidine-4-carboxamide
N-benzyl-5-(2-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
(3R,4S)-4-{4-[(3-methylthiophen-2-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
(2S,4S)-4-{4-[(1-1-benzothiophen-2-yl-N-methylformamido)methyl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
N-cyclohexyl-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-(prop-2-yn-1-yl)propanamide