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N-(5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazol-7-yl)acetamide
N-[2-(2,4-difluorophenyl)-1-[1-(2-methylbutanoyl)piperidin-4-yl]ethyl]-N-methylpropanamide
3-[4-(2-chlorophenyl)-3-oxopiperazine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinoline-2,5-dione
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-5-methylpyrazine-2-carboxamide
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-3-methyl-1-(prop-2-en-1-yl)-1H-pyrazole
2-cyclopropyl-N-(3-ethoxypropyl)-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-[(2-methoxyphenyl)methyl]-N-methyl-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
8-(1-aminocyclopropanecarbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
8-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
4-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-5-(3-fluorophenyl)-2-(trifluoromethyl)pyrimidine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methylbenzamide
(3R,4R)-1-(3-chloro-4-fluorobenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-methyl-2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethane-1-sulfonamide
N,N-dimethyl-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidine-1-sulfonamide
4-oxo-N-[2-(propan-2-yl)phenyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
(2S)-2-{[4-methyl-3-(2-oxoimidazolidin-1-yl)phenyl]formamido}-3-phenylpropanamide
(3S,4R)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-(1-ethylpiperidin-4-yl)-N-[2-(pyridin-2-yl)ethyl]oxane-2-carboxamide
N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)-1H-imidazole-5-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
N-(2,4-dimethoxyphenyl)-3-{1-[2-(2-fluorophenyl)acetyl]piperidin-4-yl}propanamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(1H-indol-4-ylmethyl)benzamide
5-fluoro-2-{1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2,6-dimethoxybenzamide
3-(furan-2-ylmethyl)-5-[1-(3-methyl-2-oxopentanoyl)piperidin-4-yl]-5-propylimidazolidine-2,4-dione
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-[1-(furan-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
methyl 5-{[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]amino}-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-phenylpiperidin-4-ol
5-benzoyl-N-cyclopropyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)[(4-methyl-1H-imidazol-5-yl)methyl]amine
(2S)-3-methyl-2-(quinoxalin-5-ylformamido)butanamide
4-benzyl-4-(hydroxymethyl)-N-(4-methoxyphenyl)piperidine-1-carboxamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
2-(1-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}ethyl)phenol
1-cycloheptyl-4-[(propan-2-yl)amino]pyrrolidin-2-one
6-(but-2-ynoyl)-N-[2-(cyclohex-1-en-1-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
5-{3-[2-(5-phenylthiophen-2-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,3,4-tetrazole
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-[(3,4,5-trimethoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-methyl-4-phenyl-3-{1-[3-(pyridin-3-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-chloro-4-fluorophenoxymethyl)-N-[2-(pyridin-4-yl)ethyl]-1,3-oxazole-4-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-5-[2-(4-methoxyphenyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-3-propanamidobenzamide
3-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-1-[2-(methylsulfanyl)phenyl]urea
N-(1-cyclopropanecarbonylpiperidin-3-yl)-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
4-benzyl-3-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}acetamide
(1S,5R)-3-(pyridin-3-ylmethyl)-6-(pyrrolidine-1-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]butane-1,2-dione
4-(3-methoxypropyl)-11-{[(3,4,5-trifluorophenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one