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N-(1-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
3-(2-chloro-6-methylphenyl)-1-(3-methoxypropyl)-1-(1-methylpiperidin-4-yl)urea
N-[1-(1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
4-[(2,5-dimethoxyphenyl)methyl]-9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 1-[(2H-1,3-benzodioxol-5-yl)carbamoyl]-3-[(2,4-difluorophenyl)methyl]piperidine-3-carboxylate
methyl[(1-{1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]amine
2-(3-methoxypropyl)-8-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-2,8-diazaspiro[4.5]decan-3-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[furan-2-yl(phenyl)methyl]acetamide
3-(1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperidin-4-yl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-4-methyl-1H-imidazole
(1R,3S,5S)-N-cyclohexyl-N-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-8-methyl-8-azabicyclo[3.2.1]octan-3-amine
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(trifluoromethyl)pyridine
6-methyl-5-{2-oxo-2-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[4-(4-{[2-(3-methoxyphenyl)ethyl]amino}piperidin-1-yl)phenyl]-2,4-dimethylbenzamide
(1S,6R)-9-[6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
4-{[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]methyl}-2-chloro-6-methoxyphenol
methyl 2-(1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
methyl (1R,3S,3aR,6aS)-3-(3-hydroxy-4-methoxyphenyl)-5-methyl-1-(2-methylpropyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
3-(2,3-dihydro-1H-isoindol-2-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]propan-1-one
1-[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-({3-[(dimethylamino)methyl]phenyl}methyl)-N,7-dimethylimidazo[1,2-a]pyridine-2-carboxamide
1-(azepan-1-yl)-3-(4-chloro-2-{[(2-hydroxyethyl)(methyl)amino]methyl}phenoxy)propan-2-ol
(3S,4S)-1-(2,5-dimethylpyrimidin-4-yl)-4-(naphthalen-2-yl)piperidin-3-ol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-[N-(4-methylphenyl)methanesulfonamido]acetamide
1-[(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-[(4-methylphenyl)methyl]pyrrolidine-2-carbonyl]-4-(1-methylpiperidin-4-yl)piperazine
4-{1-benzyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-5-methyl-1-propyl-1H-pyrazole
N-(2H-1,3-benzodioxol-5-yl)-1-(5-phenoxyfuran-2-carbonyl)piperidin-3-amine
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-[1-(3-phenylpropyl)piperidin-4-yl]-N-[3-(propan-2-yloxy)propyl]piperidine-4-carboxamide
3-(6-methoxypyridazin-3-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-methyl-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]acetamide
4-benzyl-3-ethyl-1-[3-(pyridin-3-yl)propanoyl]-1,4-diazepan-5-one
1-{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(1-{2-[1-(propan-2-yl)piperidin-4-yl]acetyl}piperidin-3-yl)benzoic acid
1-(1H-indazol-5-yl)-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperazin-2-one
5-{2-[4-(2-methoxyphenyl)piperidin-1-yl]-2-oxoethyl}-1,3-dimethylimidazolidine-2,4-dione
[2-({4-[(2-chloro-6-fluorophenyl)methyl]piperazin-1-yl}methyl)phenyl]methanol
2-[2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-5,6-dimethylpyridine-3-carbonitrile
(3S,4R)-1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-4-phenylpyrrolidine-3-carboxylic acid
4-[(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-3-yl)methyl]morpholine
5-(cyclohex-3-ene-1-carbonyl)-3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-(3-phenylpropyl)-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
methyl(naphthalen-1-ylmethyl)[(3-{2-[4-(1,3-thiazole-5-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
2-amino-6-(2,5-dimethylthiophen-3-yl)-4-[2-(ethylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
1-[2-(cyclohexylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N,N-dimethylpiperidine-4-carboxamide
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-3-(diphenylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
{4-[(2-fluoro-4-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}(pyridin-4-yl)methanol
2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol