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4-{[(3S,4R)-3-carboxy-4-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
ethyl 4-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
N-({7-[2-(4-acetylphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide
4-methoxy-6-[3-(2-methoxybenzoyl)piperidin-1-yl]pyrimidine
1-[1'-(4-fluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
3-({2-[1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
3-[(3S,4R)-1-benzyl-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(2-methoxyethyl)propanamide
1-[cyclohexyl(methyl)amino]-3-[4-({[3-(dimethylamino)propyl](methyl)amino}methyl)-2-methoxyphenoxy]propan-2-ol
1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-N-{[2-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
2-{5-[1-(1-methylpiperidin-4-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]thiophen-2-yl}pyridine
(3aR,6aS)-5-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
4-[1-(3-fluoro-4-methoxybenzoyl)piperidin-4-yl]-5-[(1E)-prop-1-en-1-yl]-2-(pyridin-3-yl)pyrimidine
(2R)-2-amino-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2-(thiophen-2-yl)acetamide
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(piperidin-4-yl)piperidine
1-(furan-2-carbonyl)-4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,4-diazepane
5-methanesulfonyl-N,2-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
2-cyclopentyl-1-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}ethan-1-one
7-(2-phenylethyl)-2-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decane
ethyl 4-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)piperidine-1-carboxylate
1-[(2-chlorophenyl)methyl]-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-4-(thiophen-2-yl)butan-1-one
(3S,4S)-4-(3-methoxyphenyl)-1-(quinolin-2-ylmethyl)piperidin-3-ol
(1S,5R)-3-(1H-indole-2-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S)-3-ethyl-4-[3-(piperidine-1-carbonyl)pyrazine-2-carbonyl]morpholine
3-(5-{3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]propanoyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
propan-2-yl 4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carboxylate
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
4-(2-methoxyethyl)-3-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-4H-1,2,4-triazole
(4aS,7aR)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N'-cyclooctyl-N-(4-hydroxybutyl)butanediamide
4-(1-{[4-(methylsulfanyl)phenyl]methyl}azetidin-3-yl)morpholine
1-ethyl-5-{[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-methyl-N-(1,2-oxazol-5-ylmethyl)-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}(methyl)(oxan-4-ylmethyl)amine
N-[(3R,4R)-4-hydroxypiperidin-3-yl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-[2-methyl-1-(pyridin-2-yl)propyl]-4-(trifluoromethyl)pyrimidin-2-amine
4-(piperidin-3-yl)-N-[4-(pyrrolidin-1-yl)butyl]benzamide
N-{1-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-1-methylpiperidine-4-carboxamide
4-[(2R)-3-hydroxy-2-{[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]amino}propyl]phenol
1-{3-[4-(trifluoromethyl)phenyl]propyl}-1H-imidazole
N-[(4-fluorophenyl)methyl]-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-(piperidine-1-carbonyl)benzene-1-sulfonamide
2-amino-6-(4-hydroxyphenyl)-4-(quinolin-4-yl)pyridine-3-carbonitrile
1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-(3-methoxyphenyl)ethan-1-one
2-(1-ethyl-1H-pyrazol-4-yl)-7-fluoro-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]quinoline-4-carboxamide
1-(2,4-dimethoxyphenyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-propylurea
1-[(1r,4r)-4-hydroxycyclohexyl]-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[4-(azepan-1-yl)butyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(4aS,8aR)-6-[3-(3-fluorophenyl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(morpholin-2-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one