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3-(4-methoxy-3,5-dimethylbenzoyl)-1-(oxan-4-yl)piperidine
5-ethyl-4-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}pyrimidin-2-amine
(4aR,7aS)-1-(cyclopropylmethyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1,3-thiazole-4-carboxamide
(3S,9aR)-3-(4-aminobutyl)-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-[1-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]pyrimidin-4-ol
4-(4-oxo-7-{spiro[2.3]hexane-1-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-[(dimethylsulfamoyl)amino]benzene-1-sulfonamide
(2S,4R)-1-{[5-(2-chlorophenyl)furan-2-yl]methyl}-N-(2-phenylethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
2-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-({7-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
1-{2-[(6,7-dimethoxy-4-methylquinolin-2-yl)amino]ethyl}imidazolidin-2-one
1-[(2,4-dimethylphenyl)methyl]-4-(2-methoxyethyl)-1,4-diazepan-5-one
1-(carbamoylmethyl)-N-{2-[(4-methylphenyl)sulfanyl]ethyl}piperidine-3-carboxamide
N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
1-[3-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-oxopropyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
6-methyl-5-{2-oxo-2-[2-(pyridin-2-yl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(2-methoxyphenyl)propanamide
(2S,4R)-4-amino-1-[2-(azepan-1-yl)-2-oxoacetyl]-N,N-diethylpyrrolidine-2-carboxamide
N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]-2-[(4-oxo-3,4-dihydroquinazolin-2-yl)sulfanyl]propanamide
N-[(4-methyl-1H-imidazol-5-yl)methyl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(pyridin-4-yl)propan-1-one
N-[3-(4-methylpiperazine-1-carbonyl)-5-({[(3-phenoxyphenyl)methyl]amino}methyl)phenyl]acetamide
methyl (2S)-2-{3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamido}-2-phenylacetate
(2S)-N2-[4-(3-fluorophenyl)phenyl]-N1-(2-methoxyethyl)pyrrolidine-1,2-dicarboxamide
3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(diphenylmethyl)propanamide
5-[4-(aminomethyl)piperidin-1-yl]-2-[(2-ethyl-1,3-thiazol-4-yl)methyl]-2,3-dihydropyridazin-3-one
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(2S)-2-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-3-hydroxypropanamide
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
(1S,5R)-6-[5-(methoxymethyl)furan-2-carbonyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[3-(furan-2-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[4-(furan-2-yl)phenyl]-3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-(2-methylphenyl)piperazin-1-yl]ethan-1-one
3-(1-methyl-1H-pyrazol-4-yl)-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}propanamide
N-methyl-2-[1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]acetamide
N-(3,4-difluorophenyl)-6-(furan-3-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
1-{2-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octane-8-carbonyl]phenyl}-1,3-diazinane-2,4-dione
1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
N-methyl-5-oxo-N-(2-phenoxyethyl)-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
(2S)-3-(4-hydroxyphenyl)-2-[(5-methanesulfonyl-2-methylpyrimidin-4-yl)amino]propanamide
6-ethoxy-2-{4-[4-(2-methoxyethoxy)piperidin-1-yl]azepan-1-yl}-4-methylquinazoline
(4aS,7aR)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1-ethylpiperidin-3-yl)methyl]-N-methyl-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)acetamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-hydroxypiperidin-1-yl)acetamide
N-[2-(4,6-dihydroxypyrimidin-2-yl)ethyl]-2,3,6-trimethylquinoline-4-carboxamide