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8-[(2-oxo-1,3-oxazolidin-5-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
[1-(azepan-1-yl)propan-2-yl]({[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl})amine
N-(2-fluoro-5-methylphenyl)-2-{[(2-methyl-1H-indol-5-yl)methyl]amino}acetamide
(2S,4S)-4-amino-1-{6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-{[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
2-(4-chlorophenoxy)-1-[1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]ethan-1-one
4-({methyl[(1-methyl-5-oxopyrrolidin-3-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
(4aS,7aR)-1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-(1-methanesulfonylpiperidin-4-yl)pyrrolidin-2-yl]pyridine
1-[4-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
ethyl 1-(5-methoxyfuran-2-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
3-{[1-(2-fluorophenyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
N-benzyl-N-(2-hydroxyethyl)-1-{2-[2-(2-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
3-(but-2-yn-1-yl)-5-[1-(3-fluorobenzoyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
methyl 1-[(3R,5S)-1-(furan-3-ylmethyl)-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
4-methyl-N-[(4-methylphenyl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-[(2,4-dimethylphenyl)methyl]-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(7-{[3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]oxolane-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-[(4-methylpiperazin-1-yl)methyl]benzamide
2-ethyl-5-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-4-methyl-1,3-oxazole
2-{4-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
3-benzyl-8-{[4-(furan-2-yl)phenyl]methyl}-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzonitrile
7-[(3,4-difluorophenyl)methyl]-2-(2,2-dimethylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
3-(1-butyl-1H-imidazol-2-yl)-1-(3,4-dimethoxybenzoyl)piperidine
1-(cyclohexylmethyl)-3-cyclopropyl-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazole
N-(2-methoxyethyl)-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-(thiophen-2-ylmethyl)acetamide
1-benzyl-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-6-hydroxy-1,4-diazepan-2-one
methyl 2-{[3-(3-chlorobenzoyl)piperidine-1-carbonyl]amino}benzoate
(2S,4R)-4-amino-N-methyl-1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carbonyl]pyrrolidine-2-carboxamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-(4-phenyl-1,4-diazepan-1-yl)ethan-1-one
methyl 1-(2-methoxyethoxy)-8-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(methyl){[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-N-(pyridin-4-ylmethyl)-4-(trifluoromethyl)benzene-1-sulfonamide
3,3,3-trifluoro-2-hydroxy-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]propanamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-methylpiperidine-2-carboxamide
1-(1H-pyrazole-4-carbonyl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
5-({2-[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,3-triazole
1-(5-tert-butyl-2-methoxyphenyl)-3-{2-[(2R)-pyrrolidin-2-yl]ethyl}urea
[(3R,4R)-1-[(2-methylnaphthalen-1-yl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-(dimethylamino)-4-methyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]pyrimidine-5-carboxamide
2-cyclopentyl-4-[4-(2-methoxy-2-phenylacetyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(but-2-yn-1-yl)-5-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
2-cyclohexyl-N-(2-hydroxy-2-phenylethyl)-N-methyl-1,3-benzoxazole-6-carboxamide
N-cycloheptyl-1-cyclopropyl-5-[3-(diethylcarbamoyl)piperidine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
6-[(cyclopropylmethyl)amino]-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]pyridine-3-carboxamide
N-[(4-ethylphenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methylazepan-4-amine