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1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
9-[(5-fluoro-2-methylphenyl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(5-phenyl-4H-1,2,4-triazol-3-yl)ethan-1-one
N,N-dimethyl-2-phenyl-7-{spiro[2.3]hexane-1-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(4-{[4-(1-benzylpiperidine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-ol
N-[(2-hydroxypyridin-3-yl)methyl]-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
(3S,4S)-1-{[3-(furan-2-yl)phenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-(4-methoxyphenoxy)ethan-1-one
1-cyclopropyl-N-methyl-6-oxo-N-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
3-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
2-{3-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]propyl}-1,3-benzothiazole
5-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
N-methyl-N-(2-phenylethyl)piperidin-3-amine
5-[2-(cyclohex-1-en-1-yl)acetyl]-N-cyclopropyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3-(2-fluorophenyl)-3-phenylpropanamide
2-({[1-(3,5-dimethyladamantane-1-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
methyl 1-[(3R,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[3-(1H-indol-2-yl)phenyl]-1-(5-methoxyfuran-2-carbonyl)piperidine-3-carboxamide
2-(3-methoxypropyl)-8-[2-(thiophen-3-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)(oxolan-3-ylmethyl)amine
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
4-{[6-(2,3-difluorophenyl)pyridin-3-yl]methyl}morpholine
4-[1-(2,3-difluorobenzoyl)piperidin-3-yl]-5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidine
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzamide
1-(2-methoxy-4-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
methyl 2-[2-oxo-4-(thiophene-3-carbonyl)piperazin-1-yl]acetate
[2-(2-methoxy-6-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}phenoxy)ethyl]dimethylamine
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
1-(4,7-dimethylquinazolin-2-yl)-N-[(4-phenyloxan-4-yl)methyl]piperidine-4-carboxamide
8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2-aminopyrimidin-5-yl)methyl]-1-methyl-3-(3,4,5-trimethoxyphenyl)urea
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]acetamide
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-(pyridin-4-ylmethyl)propanamide
methyl 8-[(2,3-dimethoxyphenyl)methyl]-1-(3-methylbutoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
6-methyl-N-[2-(morpholin-4-yl)ethyl]-2-propylpyrimidin-4-amine
2-{1-benzyl-4-[(1-methyl-1H-indol-3-yl)methyl]piperazin-2-yl}ethan-1-ol
8-(5-fluoro-1H-indole-2-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(1-ethyl-1H-indazol-3-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
5-fluoro-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}quinazolin-4-amine
2-(dimethylamino)-2-(2-fluorophenyl)-1-(pyrrolidin-1-yl)ethan-1-one
8-(1,3-benzothiazol-2-ylmethyl)-1-ethyl-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2-fluorophenyl)methoxy]-8-[2-(4-methylphenoxy)acetyl]-1,8-diazaspiro[4.5]decan-2-one
N-{[1-(9H-fluoren-2-ylmethyl)piperidin-3-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxamide
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
N-methyl-3-(1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-3-yl)-N-(1-methylpiperidin-4-yl)propanamide
1-{6-methyl-5-[5-(thiophen-3-ylmethyl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}propan-1-one
(1-{5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}-2-methylpropan-2-yl)dimethylamine
5-(2-chloro-4-fluorophenoxymethyl)-N-[(2-methylphenyl)methyl]-1,2-oxazole-3-carboxamide