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N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-[5-(2-methyl-1,3-thiazol-4-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N,N-diethyl-2-({1-[(4-methoxyphenyl)methyl]-2-oxo-4-(pyridin-3-ylmethyl)-1,4-diazepan-6-yl}oxy)acetamide
3-{1-[(1,2-dimethyl-1H-indol-3-yl)methyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
3-{4-[(2,2-diphenylcyclopropyl)methyl]piperazin-1-yl}propanamide
8-[(4-ethoxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-4-phenylpiperidin-4-ol
9-(2,6-dimethylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-(1,2-diphenylethyl)propanamide
2-[(4aR,8aS)-6-(4-fluorobenzoyl)-decahydro-1,6-naphthyridine-1-carbonyl]-N,N-dimethylaniline
5-[(2,6-difluorophenyl)methyl]-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}quinoxaline
N-{[7-(2-chloro-4-fluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-2-(morpholin-4-yl)benzamide
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}acetamide
3-(2-ethylbutyl)-8-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(4-cyclohexylpiperazine-1-carbonyl)-1-methyl-1H-pyrrole-3-carbonitrile
1-(cyclopropylmethyl)-3-({[(3-fluoro-4-methylphenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
4-(2,2-diphenylethyl)-3-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
2,2-dimethyl-1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-4-(pyridin-3-yl)piperazine
2-{4-[2-(2-oxopyrrolidin-1-yl)propanoyl]piperazin-1-yl}benzonitrile
(5-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1H-1,3-benzodiazol-2-yl)methanol
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(1-methyl-1H-imidazole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-(3-phenylpropyl)piperidin-3-amine
(1S,4S)-5-(6-ethylpyrimidin-4-yl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-3-yl]methyl}-4-fluorobenzamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
5-[3-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)propyl]-1,3,4-thiadiazol-2-amine
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)-4-methyl-1,2,5-oxadiazole-3-carboxamide
(1-methyl-1H-imidazol-2-yl)(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)methanol
9-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
8-[(4-methoxy-3-methylphenyl)methyl]-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]-1H-indazole-3-carboxamide
N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
N-(1,3-dihydroxy-2-methylpropan-2-yl)-2-(5,6,7,8-tetrahydronaphthalen-2-yloxy)butanamide
N-{1-[1-(2-cyclohexylacetyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxy-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]piperidine-1-carboxamide
6-{[4-(hydroxydiphenylmethyl)piperidin-1-yl]methyl}-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
[(3R,4R)-1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-3-{2-oxo-2-[4-(piperidin-1-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
methyl 5-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N-cyclopropylfuran-2-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(pyridin-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aS,8aR)-6-(2-cyclopropylpyrimidine-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
9-[(3-chloro-4-ethoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one