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5-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidine-1-carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate
N-{[2-(2-cyclobutaneamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,5-dimethoxybenzamide
5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-benzotriazole
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-methyl-1H-pyrazole-3-carboxamide
2-{[2-(pyridin-3-yl)-1,3-thiazol-4-yl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperidin-4-ol
4-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}acetamide
2-(piperidin-1-ylmethyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]-1,4-oxazepane
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
3-methyl-7-[3-(3-methylpiperidin-1-yl)-3-oxopropyl]-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
6-tert-butyl-N-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-(cyclopropylmethyl)-6-(2,5-dimethylfuran-3-yl)-N-(2-fluoroethyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(4-fluorophenyl)-4-(5-propyl-1,2-oxazole-4-carbonyl)-1,4-diazepane
N,5,6-trimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidin-4-amine
N-[2-(1-cyclopentylpiperidin-4-yl)ethyl]oxolane-3-carboxamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
8-fluoro-3-[(5-oxopyrrolidin-2-yl)methyl]-3,4-dihydroquinazolin-4-one
3-(4-methylpiperazine-1-carbonyl)-N-[(1-phenylcyclopentyl)methyl]-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(3-methylphenyl)-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-{2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
2-butyl-4-{[4-(5-methylfuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
N-methyl-N-(1-methylpiperidin-4-yl)-3-[1-(4-oxo-4-phenylbutanoyl)piperidin-3-yl]propanamide
2-[methyl({4-methyl-5-[1-(9H-purin-6-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
(3R,5S)-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
5-(2-methoxyphenoxymethyl)-N-methyl-N-(2-methylpropyl)-1H-pyrazole-3-carboxamide
2-methyl-4-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-(3-{4-[(2-acetamido-3-methylbutanamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)-5-methylthiophene-2-carboxamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
4-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}quinazoline
3-{9-[2-(2-fluorophenyl)ethoxy]-10-(methoxycarbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-3-carbonyl}pyridin-1-ium-1-olate
1-[4-(4-chlorophenoxy)piperidin-1-yl]-3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
(3S,4S)-4-(naphthalen-2-yl)-1-(1,3-thiazole-4-carbonyl)piperidin-3-ol
N-[(1R,3R)-3-aminocyclopentyl]-8-fluoro-4-oxo-1,4-dihydroquinoline-2-carboxamide
1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}azetidin-3-ol
8-{[4-(3,3,4-trimethylpiperazine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
1-(4-chlorophenyl)-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
6-(2-aminoethyl)-2-(4-chlorophenyl)-3,4-dihydropyrimidin-4-one
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1-ethyl-4-{[3-(3-methoxypropyl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
6-{9-oxa-2-azaspiro[5.5]undecan-2-ylmethyl}pyridine-2-carboxylic acid
N-cyclohexyl-3-[4-(4-methoxyphenyl)-3-oxopiperazin-1-yl]propanamide
1-[3-(pyridin-4-yl)azetidin-1-yl]isoquinoline
N-[3-(dimethylamino)-2,2-dimethylpropyl]-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)propan-2-ol
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]acetamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-4-(quinolin-2-ylmethyl)-1,4-diazepan-2-one
methyl 1-methoxy-2-oxo-8-(3-phenylpropyl)-1,8-diazaspiro[4.5]decane-4-carboxylate