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4-(5-chloro-2-fluorobenzoyl)-6-methoxy-1-[(4-methoxyphenyl)methyl]-1,4-diazepan-2-one
5-ethyl-4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methylpyrimidine
2-{[butyl(methyl)amino]methyl}-4-(7-chloroquinolin-4-yl)phenol
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
2-benzyl-N-[(3-methylpyridin-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
4-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-ethyl-6-methyl-N4-[2-(4-methyl-1H-imidazol-2-yl)ethyl]pyrimidine-2,4-diamine
N-[(2R,4R,6S)-2-cyclohexyl-6-(2-phenyl-1,3-oxazol-4-yl)oxan-4-yl]acetamide
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-3-(1H-pyrazol-4-yl)propanamide
N-[2-(ethylsulfanyl)phenyl]-4-(4-methoxypyrimidin-2-yl)piperazine-1-carboxamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)(pyridin-2-ylmethyl)amine
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(trifluoromethyl)pyridin-2-amine
2-[4-(5-ethyl-2-methylpyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
N,2,5-trimethyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
7-methoxy-3-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carbonyl)-2,3,4,5-tetrahydro-1H-3-benzazepine
2-(2,3-difluorophenoxymethyl)-N-[2-(6-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
2-ethyl-8-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(3S,4R)-1-(1H-pyrazole-4-sulfonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
[(5-chloro-2-methoxyphenyl)methyl](ethyl)(1,3-thiazol-2-ylmethyl)amine
N-benzyl-2-{[(cyclopropylmethyl)amino]methyl}-N-methyl-2,3-dihydro-1H-inden-2-amine
1-(3-methylpyridin-4-yl)-4-[3-(methylsulfanyl)propyl]piperazine
1-(2-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)pyrrolidin-2-one
1-[7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(4-hydroxyphenyl)-2-phenylpropan-1-one
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2-(2,3,6-trifluorophenyl)acetamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]hexan-1-one
3-(2-chlorophenyl)-N-{[5-methyl-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
N-({5-[(1,4-dimethylpiperidin-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-(1-{7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-methoxy-N-methylbenzamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
N4-(2,3-dihydro-1H-inden-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-[1-(pyrimidin-5-ylmethyl)piperidin-3-yl]benzoic acid
1-{2-[3-(2-methoxybenzoyl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-2,4-dimethoxypyrimidine
N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(trifluoromethyl)benzamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[(5-fluoro-1H-indol-2-yl)methyl]-3-(2-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](ethyl){[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-ethyl-N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-6-oxopiperidine-3-carboxamide
1-(4-chlorophenyl)-N-{[5-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropane-1-carboxamide
1-[7-(1,3-benzothiazol-2-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
2-{5-[5-(hydroxymethyl)furan-2-yl]-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
4-(8-methylquinolin-5-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-1-yl)-1-phenylethyl]amine
1-[5-methoxy-2-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
1-cyclopentyl-5-(pyrrolidine-1-carbonyl)piperidin-2-one
(4aS,8aR)-6-[6-(dimethylamino)pyrazin-2-yl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(2R,3R)-2-(benzyloxy)-1'-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
(1S,5R)-3-[2-chloro-5-(trifluoromethyl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one