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methyl({[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
[3-(3-phenylpropyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl]methanol
cyclopentyl 4-{[methyl({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})carbamoyl]amino}benzoate
5-[(2S)-1-cyclohexanecarbonylpyrrolidin-2-yl]-1-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazole
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-methylfuran-2-carbonyl)piperidin-3-ol
5-(2-fluoro-6-methoxyphenoxymethyl)-3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazole
(2S,4R)-4-amino-N-ethyl-1-[2-(2-methoxyphenoxy)acetyl]pyrrolidine-2-carboxamide
2-cyclohexyl-5-{[4-(2-methylpyridin-4-yl)piperazin-1-yl]methyl}pyrimidine
6-(4-fluorophenyl)-2-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}pyridine-3-carboxylic acid
2-{4-[(2,3-difluorophenyl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
2-{1-[(3,4-difluorophenyl)methyl]-4-(isoquinolin-5-ylmethyl)piperazin-2-yl}ethan-1-ol
1-(morpholin-4-yl)-3-[5-(1H-pyrrole-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propan-1-one
2-(2,3-difluorophenyl)-2-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}acetic acid
N-[(3-fluorophenyl)methyl]-5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
(4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-oxazepan-6-yl)methanol
1-(4-fluorophenyl)-4-(piperidin-3-yl)piperazine
N-cyclopropyl-1-{1-[(2E)-3-(2,3-difluorophenyl)prop-2-enoyl]piperidin-4-yl}piperidine-4-carboxamide
4-{1-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl}pyridine
(1S,5R)-3-(pyrimidin-2-yl)-6-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
methyl({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})[1-(pyridin-3-yl)ethyl]amine
3-cyclopropyl-5-[1-(methoxymethyl)cyclobutyl]-1-(4-methoxyphenyl)-1H-1,2,4-triazole
3-cyclopentyl-5-[(oxolan-2-ylmethoxy)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1,3,7-trimethyl-1H-indole-2-carboxamide
3-{[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}-2-(thiophen-3-ylmethyl)propan-1-ol
N-(1,4-dioxan-2-ylmethyl)-N-methyl-3-[4-(piperidin-1-yl)piperidine-1-carbonyl]-6-(thiophen-2-yl)pyridin-2-amine
N-methyl-3-{[2-(pyridin-2-yl)-1H-imidazol-1-yl]methyl}benzamide
ethyl 2-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
1-amino-N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]cyclopropane-1-carboxamide
1-[(4aR,8aR)-4a-hydroxy-7-[(2-methyl-1-benzothiophen-3-yl)methyl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
2-methyl-4-{4-[7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}but-3-yn-2-ol
methyl 3-[(4-methoxy-3-methylphenyl)methyl]-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4,5-dimethyl-6-[4-(thiomorpholin-4-yl)piperidin-1-yl]pyrimidin-2-amine
methyl 4-({[2-(1-butyl-5-oxopyrrolidin-2-yl)ethyl]amino}methyl)benzoate
N-[(2-ethoxypyridin-3-yl)methyl]-6-(methoxymethyl)pyrimidin-4-amine
6-(3-chlorophenyl)-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-N-(propan-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
9-methoxy-7-oxo-3-(3-phenylpropanoyl)-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
9-(5,6-dimethylpyrimidin-4-yl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-3-[(dimethylamino)methyl]pyrrolidin-3-ol
4-hydroxy-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-phenylpyrimidine-5-carboxamide
N,N-diethyl-3-{[1-(4-methyl-1H-imidazol-2-yl)propyl]sulfamoyl}benzamide
5-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methylpyridine
8-(2,2-dimethylpropyl)-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(1,4-oxazepan-4-ylmethyl)phenyl]-6-(oxolan-3-yl)-3,4-dihydropyrimidin-4-one
1-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]urea
6-benzyl-N-(3,4-difluorophenyl)-6-azaspiro[2.5]octane-1-carboxamide
3-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
(3S,4S)-1-[(6-ethoxypyridin-3-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-cyclopentyl-1-(2-methylpropyl)-5-(2-phenoxypropanoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(1-methyl-1H-imidazol-2-yl)-1-(pyrrolidine-1-sulfonyl)piperidine