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N-[2-(2,4-dichlorophenyl)ethyl]morpholine-2-carboxamide
5-benzamido-1-cyclopentyl-N-methyl-N-(propan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
5-[2-(furan-2-yl)-2-phenylethyl]-3-methyl-1H-1,2,4-triazole
{4-[(4-chlorophenyl)methyl]-1-(6-methoxypyrimidin-4-yl)piperidin-4-yl}methanol
[4-methyl-5-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methanol
7-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
5-{[(furan-2-ylmethyl)(prop-2-en-1-yl)amino]methyl}-2-hydroxybenzoic acid
1-[4-(pyridin-4-yl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
2-methyl-N-(1-{7-[(3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
2,5-dioxo-6-(2-phenoxyethyl)-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,5-dimethoxybenzamide
5-(2-chloro-6-methoxyphenyl)pyridine-3-carboxylic acid
4-(2,2-dimethyloxane-4-carbonyl)-7-(thianthren-1-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1S,5R)-3-[4-(2-oxopyrrolidin-1-yl)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(2,4-difluorophenyl)-1-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]ethyl]-N-methylpyridine-3-carboxamide
2-(cyclopent-2-en-1-yl)-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide
N-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-4-(2-fluorophenyl)piperazine-1-carboxamide
N-({4-[(3,5-dimethoxyphenyl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
7,7-dimethyl-N-[(5-methylthiophen-2-yl)methyl]-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
{[5-(1-benzylpiperidin-4-yl)-4-ethyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
5-{4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidine-1-carbonyl}-2-methyl-1,4-dihydropyridin-4-one
N,N-dimethyl-2-{4-[(3-phenyloxolan-3-yl)methyl]-1,4-diazepan-1-yl}acetamide
1-(4-cyanophenyl)-3-(2,2-dimethyloxan-4-yl)-3-ethylurea
4-[3-benzyl-3-(hydroxymethyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
(1-{1-[(9-ethyl-9H-carbazol-3-yl)methyl]piperidin-3-yl}piperidin-4-yl)methanol
1-(1,4-dioxan-2-ylmethyl)-5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-3-(oxan-4-yl)-1H-1,2,4-triazole
4-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(quinolin-4-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
1-cycloheptyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
8-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-2,8-diazaspiro[4.5]decan-3-one
2-[9-(5-fluoropyrimidin-2-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-(3-fluoro-4-methoxyphenyl)-N-methyl-1,2,4-triazin-3-amine
8-(2-ethylbutyl)-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]methanol
2-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]pyridine-3-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(3-methylpyridin-2-yl)ethyl]piperidine-3-carboxamide
2-({2-[3-(furan-2-yl)phenyl]-1H-imidazol-1-yl}methyl)-5-methylpyrazine
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-3-carboxamide
1-cycloheptyl-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-oxopiperidine-3-carboxamide
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5-methylpyrazine
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-7-fluoro-2-methylquinoline-4-carboxamide
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
ethyl 4-(oxan-2-ylmethyl)-1-[2-(phenylsulfanyl)acetyl]piperidine-4-carboxylate
5,6-dimethyl-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}pyrimidin-4-amine
dimethyl({4-methyl-5-[1-(4-methylquinolin-2-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
methyl 1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-(3-{4-[(2,2-dimethyloxan-4-yl)amino]piperidin-1-yl}phenyl)imidazolidin-2-one
N-(2H-1,3-benzodioxol-5-yl)-3-(2,3-dimethoxyphenyl)pyrrolidine-1-carboxamide