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6-fluoro-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-1,3-benzodiazole-2-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]azepane-4-carboxamide
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]urea
2-(1-{[1-(3-methylquinolin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
2-methoxy-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pyridine-4-carboxamide
1-(morpholin-4-yl)-3-[3-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]propan-2-ol
N-{1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-4-yl}pyrimidin-2-amine
2-(2-methyl-1,3-thiazol-4-yl)-5-(2-phenylmorpholine-4-carbonyl)pyrimidin-4-ol
2-{4-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]morpholin-3-yl}acetic acid
(3aS,6aS)-1-(3,4-dimethoxybenzenesulfonyl)-octahydropyrrolo[2,3-c]pyrrole
methyl 5-{[(3-chlorophenyl)methyl]amino}-3-(furan-2-amido)-1-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]propane-1,2-diol
2-(2-hydroxyethyl)-6-[4-(pyridin-3-yl)pyrimidin-2-yl]-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
4-(2,4-dimethylpyrimidine-5-carbonyl)-1-(3-methoxyphenyl)-5-methylpiperazin-2-one
2-ethyl-6-[4-(4-fluorophenyl)oxane-4-carbonyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-[(6-chloropyridin-3-yl)methyl]-4-(2,2-dimethoxyethyl)piperazine
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
N,N-diethyl-5-methyl-4-[(2-phenylethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
5-cyclobutanecarbonyl-1'-[3-(methylsulfanyl)butyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(furan-2-ylmethyl)-4-(3-propoxypiperidine-1-carbonyl)piperidine
2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(prop-2-en-1-yl)acetamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidine
2-[2-(3,4-diethoxyphenyl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-{3-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-(naphthalen-2-ylmethyl)pyrrolidin-2-one
2-{2-[2-(trifluoromethyl)benzoyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
3-(2,5-difluorobenzoyl)-1-(3-methylthiophene-2-carbonyl)piperidine
N,N-dimethyl-2-{[2-(4-methyl-1H-pyrazol-1-yl)propanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
ethyl 2-(1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)acetate
1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyrrolidin-1-yl)piperidine
1-[3-(1H-pyrazol-1-yl)benzoyl]-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
3,5-difluoro-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-methyl-6-oxo-4-(6-phenoxypyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(2-methylphenyl)piperidine
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
4-chloro-1-methyl-3-{[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]methyl}-1H-indazole
1-(4-{5-[(4-acetylpiperazin-1-yl)methyl]-2-methoxyphenoxy}piperidin-1-yl)-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-(2-ethoxyphenyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
(1S,5R)-6-[(4-methoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(oxolan-2-ylmethyl)-9-[3-(thiophen-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
5-({4-phenyl-5-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-1H-1,2,4-triazole
2-(2-{[2-(1H-imidazol-4-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-(benzyloxy)-1-{3-[(3-methoxyphenyl)methyl]-1,2-oxazole-5-carbonyl}piperidine
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(5-ethyl-2-methylpyrimidin-4-yl)pyrrolidine-3-carboxylic acid
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
1-(2-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one