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2-(morpholin-3-yl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]acetamide
N-(3-cyclopentylpropyl)-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-methoxy-2-{[7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
9-(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinoline-3,7-dione
(4aR,8aR)-2-[(5-propylfuran-2-yl)methyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
ethyl 3-[(3-methoxyphenyl)methyl]-1-[2-(methylsulfanyl)acetyl]piperidine-3-carboxylate
N,1,3-trimethyl-N-(1-{1-[(4-oxo-4H-chromen-3-yl)methyl]piperidin-4-yl}-2-phenylethyl)-1H-pyrazole-5-carboxamide
8-[(2-ethylphenyl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,1-dimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
ethyl 4-[4-(5-methylfuran-2-yl)benzamido]piperidine-1-carboxylate
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-difluorobenzamide
4-(1H-pyrazol-1-yl)-1-(pyrrolidine-1-carbonyl)piperidine-4-carboxylic acid
4-(1-butyl-1H-pyrazol-4-yl)-1-[2-(piperidin-1-yl)ethyl]-1,2,3,6-tetrahydropyridine
N-[2-(3,4-dimethoxyphenyl)ethyl]-3-(4-methoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}piperidine-4-carboxamide
1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-(morpholin-4-yl)-2-[4-(1-phenyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethan-1-one
5-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
2-(4-{[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
2,2-dimethyl-N-(1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1-hydroxycyclopentane-1-carboxamide
1-cyclopentyl-3-(2-methylphenyl)-3-[2-(morpholin-4-yl)-2-oxoethyl]pyrrolidine-2,5-dione
N-(4-fluorophenyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperazine-2-carboxamide
4-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-2-(propan-2-yl)-N-(pyridin-2-ylmethyl)-1,3-thiazole-5-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methylimidazo[1,2-a]pyridine-6-carboxamide
2-[2-(morpholin-4-ylmethyl)-4-(pyrazin-2-yl)phenoxy]-N-(quinolin-3-ylmethyl)acetamide
N4-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)morpholine-2,4-dicarboxamide
N-ethyl-3-[(2-methoxyethyl)(methyl)sulfamoyl]-N-(oxan-4-yl)benzamide
1-(5-chloro-2-ethyl-3-methyl-1-benzofuran-7-yl)-3-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]urea
(1S,5R)-6-benzyl-3-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
6-{[(4-fluorophenyl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-(furan-2-ylmethyl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}piperidine-3-carboxamide
(2E)-N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3-phenylprop-2-enamide
3-chloro-N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2,3-dihydro-1H-inden-2-yl)acetamide
3-[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1-methyl-1,2-dihydroquinoxalin-2-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-cyclobutyl-N,1-dimethyl-7-(oxolane-2-amido)-1H-1,3-benzodiazole-5-carboxamide
N-{1-[4-(3,4-dihydro-2H-1,4-benzoxazine-4-carbonyl)phenyl]-1H-pyrazol-4-yl}-2-(3-fluorophenyl)acetamide
1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]-4-phenylbutan-1-one
2-{1-[(2-methylphenyl)methyl]-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
1-{1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carbonyl}piperidin-4-ol
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-1-methyl-1H-pyrazole-4-carboxamide
N-{[7-(6-ethyl-2-methylquinoline-4-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(5-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}furan-2-yl)methanol
(2R)-2-amino-1-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-phenylethan-1-one
1-(azocan-1-yl)-3-(2-methoxy-5-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
2-[4-(hydroxymethyl)phenyl]-2-[methyl(1H-pyrazol-3-ylmethyl)amino]acetic acid
ethyl 2-[4-(benzylsulfamoyl)piperazin-1-yl]acetate
(5S,9aS,9bS)-5-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one