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3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(3,4,5-trimethoxyphenyl)methyl]propanamide
1-(azepan-1-yl)-3-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]propan-2-ol
4-{6-[2-(pyridin-3-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(propan-2-yl)amine
2-(4-chlorophenyl)-2-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}acetic acid
2-methyl-N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]pyridine-3-carboxamide
2-(3-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-1-[(4-methoxyphenyl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperazine
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}({[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})(2-methoxyethyl)amine
2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
3-(2-amino-1,3-thiazol-4-yl)-N-(2,3-dihydro-1H-inden-2-yl)propanamide
3-[2-methyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]propanoic acid
4-(2,3,6-trimethylquinoline-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(3-methoxyphenyl)methyl]methylamine
1-cyclohexyl-6-(pyridin-3-ylmethoxy)-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1,4-diazepan-2-one
(4aR,7aS)-1-cyclopropanecarbonyl-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-1-{[5-(4-chlorophenyl)furan-2-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
9-(3-hydroxypyridine-2-carbonyl)-4-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-2-ethyl-7-(2-methoxybenzamido)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
3-[3-(4-fluorophenyl)pyrrolidin-1-yl]-6-methylpyridazine
benzyl[(2,4-dimethoxypyrimidin-5-yl)methyl](1,3-thiazol-2-ylmethyl)amine
9-(3,5-dimethoxybenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[1-(2-oxo-4-phenylbutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
2-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
3-phenyl-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
[4-(2,1,3-benzothiadiazol-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl](2-chloro-6-fluorophenyl)methanol
3-benzoyl-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
1-(azocan-1-yl)-3-[2-methoxy-5-({[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-({7-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
3-hydroxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyridine-2-carboxamide
N-(2-methylpropyl)-3-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-sulfonyl]benzamide
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(3-fluorophenyl)acetamide
2-[benzyl(methyl)amino]-N-methyl-N-(1,2-oxazol-3-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
1-cyclopentyl-N3-methyl-N5-(2-methylpropyl)-4-oxo-N3-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-{1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-3-yl}ethan-1-one
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine
3-{2-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 9-[2-(2-fluorophenyl)ethoxy]-3-(3-methylpentanoyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(1-{1-[(1,2-dimethyl-1H-indol-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
N-({1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
4,4,4-trifluoro-1-[1-(4-methoxy-2,3-dimethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]butan-1-one
3-({1-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}methyl)benzamide
6-fluoro-4-methyl-2-{2-[4-(pyridin-2-yl)piperazine-1-carbonyl]pyrrolidin-1-yl}quinazoline
4-(2-methoxyphenoxy)-1-[(5-methylthiophen-2-yl)methyl]piperidine-4-carboxylic acid
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-4-enamide
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
1-{1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-3-phenylpropan-1-ol
N-({1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
6-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}pyrazine-2-carboxamide