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1-cyclobutanecarbonyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)piperidine-4-carboxamide
N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
{1-[(6-methylpyridin-2-yl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
1-[2-(dimethylamino)ethyl]-N-(9H-fluoren-9-yl)-5-oxopyrrolidine-3-carboxamide
8-(5-acetylpyridin-2-yl)-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-ethyl-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
N-[1-(furan-2-carbonyl)piperidin-3-yl]-6-methoxypyrimidin-4-amine
ethyl 4-[(4-{[1-(2,3-dimethyl-1H-indole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
6-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
1-(2,3-dichlorophenyl)-4-{2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}piperazine
2-amino-7-(6-chloro-2-methylquinoline-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-4-phenylbutane-1,4-dione
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-3-(1,2-oxazinan-2-yl)propanamide
3-(cyclopentylsulfamoyl)-N-(oxan-3-ylmethyl)benzamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-2-(2,4-dioxoimidazolidin-1-yl)-N-(2-hydroxyethyl)acetamide
N-[(3R,4S)-1-(cyclobutylmethyl)-4-cyclopropylpyrrolidin-3-yl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
4-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
3-[(cyclohexylamino)methyl]-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-3-(2-oxoimidazolidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
1-cyclopentyl-4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-2-one
(1S,4S)-2-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-2-azabicyclo[2.2.1]heptane
(2S)-2-[4-(6-methoxypyridin-3-yl)-1H-1,2,3-triazol-1-yl]-4-methylpentan-1-ol
N-methyl-N-(oxan-4-yl)-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]propanamide
N-methyl-2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
3-fluoro-N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-7-methylimidazo[1,2-a]pyridine-2-carboxamide
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl][(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]methylamine
N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(naphthalen-1-yl)acetamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
(3R,4S)-4-cyclopropyl-1-[4-(trifluoromethyl)benzenesulfonyl]pyrrolidin-3-amine
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}amine
3-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-1-(2-methylpropyl)-1-(pyridin-2-ylmethyl)urea
N-[3-(4-fluorophenyl)phenyl]-1-(3,3,3-trifluoropropanoyl)piperidine-3-carboxamide
5-benzenesulfonamido-1-ethyl-N-[2-(3-methoxyphenyl)ethyl]-2-methyl-1H-1,3-benzodiazole-7-carboxamide
3-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N-(pyridin-3-yl)propanamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
methyl (2S)-2-{[5-(5-methylfuran-2-yl)-1,2,4-triazin-3-yl]amino}-3-phenylpropanoate
N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-methyl-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-amine
5-[4-(2,3-dimethylphenyl)piperazin-1-yl]-1-(4-methylpentyl)azepan-2-one
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
7-(2-methoxyethyl)-2-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
(3S,4S)-1-(2,6-dimethylquinoline-4-carbonyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
N-{2-[4-({[3-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]formamido}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}pyridine-2-carboxamide
8-[(4-methyl-1H-imidazol-2-yl)methyl]-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methyl-1-[3-(2-methylphenoxy)azetidin-1-yl]-2-(morpholin-4-yl)propan-1-one
N-cyclohexyl-5,6-dimethyl-2-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
7,7-dimethyl-2-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(3-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one