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N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](1H-imidazol-2-ylmethyl)(2-methoxyethyl)amine
4-[(6-methoxypyrimidin-4-yl)amino]-1-(3-phenylpropyl)pyrrolidin-2-one
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
2-phenoxy-N-(2-{7-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
methyl 4-(5-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
2-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]-6-methylphenol
1-(3-{[4-(6-ethoxy-4-methylquinazolin-2-yl)-1,4-diazepan-1-yl]methyl}phenyl)ethan-1-one
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-hydroxy-4-(methylsulfanyl)butan-1-one
N-{1-[1-(2-oxopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
1-{4-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}-4-methylpiperazine
N-[1-(1,3-thiazol-2-yl)ethyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
1-cyclopentyl-4-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
2-[4-fluoro-3-(hydroxymethyl)phenyl]-2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]acetic acid
1-(1-cyclopropylethyl)-5-(2-ethoxyphenyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(3-methoxyphenyl)-1-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)ethyl]-N-methylfuran-2-carboxamide
(3R,4S)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
(1R,3S)-3-{[1-(phenylcarbamoyl)piperidin-4-yl]carbamoyl}cyclopentane-1-carboxylic acid
methyl (2S,4S)-4-[2-chloro-5-(trifluoromethyl)benzamido]-1-[(2-ethoxyphenyl)methyl]pyrrolidine-2-carboxylate
5-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}pyrazin-2-ol
N-(2-methoxyethyl)-2-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(2R,3S,6R)-3-(2-methoxyphenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-sulfonamide
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
7-(3-chlorophenyl)-4-(furan-2-carbonyl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aR,7aS)-1-(2-methoxyethyl)-4-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2-oxo-N-(thiophen-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-[(3-methoxyphenyl)methyl]-8-(oxane-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(2S,4S)-N-ethyl-4-[2-(2-methyl-1H-imidazol-1-yl)acetamido]-1-(pent-2-yn-1-yl)pyrrolidine-2-carboxamide
1-(propan-2-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
N-(2-hydroxy-2-phenylethyl)-2-(methoxymethyl)-N,6-dimethyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
N-[4-(5-methyl-4-{[(1-methylcyclohexyl)formamido]methyl}-1,3-oxazol-2-yl)phenyl]pyridine-3-carboxamide
N-({1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}methyl)-1H-1,2,4-triazole-5-carboxamide
N-methyl-3-[(2-oxo-1,2-dihydroquinoxalin-1-yl)methyl]-1,2,4-oxadiazole-5-carboxamide
2-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
[(3R,4R)-1-(2-methoxypyridine-3-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[2-(1,1-dioxo-1λ6-thiolan-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[2-(2-fluorophenyl)ethyl]piperidine-3-carboxamide
1-(5-{[(dimethylsulfamoyl)amino]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)-2-(thiophen-2-yl)ethan-1-one
(2,3-dihydro-1-benzofuran-5-ylmethyl)(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
N-(3-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-3-oxopropyl)acetamide
N-({1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}methyl)-4-methoxybenzene-1-sulfonamide
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-4-[3-(thiophen-2-yl)propanoyl]-1,4-diazepan-2-one
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-4-({[(1-ethyl-1H-imidazol-2-yl)methyl]amino}methyl)-2-methylpyrrolidin-2-yl]methanol
(3R,4S)-1-(4-chloro-2-fluorobenzoyl)-4-cyclopropylpyrrolidin-3-amine
N-{2-[(dimethylcarbamoyl)methyl]phenyl}-3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide
3-[(2-ethoxyphenyl)methyl]-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-cyclopropyl-N-({4-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)thiophene-2-carboxamide