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N-[(2-chlorophenyl)methyl]-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamide
5-methoxy-2-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)pyridin-4-ol
1-[4-(2-{2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethoxy)phenyl]propan-1-one
1-cyclopentyl-3-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
(3S,7S,8aS)-3-(4-aminobutyl)-7-{[(3-fluoro-4-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-benzyl-8-[(2,3-difluorophenyl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-({8-[(4-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-5-(4-methoxyphenyl)furan-2-carboxamide
(furan-3-ylmethyl)(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amine
1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]cyclopropane-1-carboxamide
(2S)-2-amino-1-[4-(4-chlorophenoxy)piperidin-1-yl]-4-(methylsulfanyl)butan-1-one
2-(2H-1,3-benzodioxol-5-yl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}acetamide
methyl 3-{[3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
1-[1-(2-aminopyridine-4-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
(2E)-N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methylpent-2-enamide
1-(3-fluoro-4-methoxybenzoyl)-4-(1H-imidazol-2-yl)piperidine
dimethyl(1-{3-[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]phenyl}ethyl)amine
1-{4-[2-(aminomethyl)morpholin-4-yl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(1H-pyrazol-1-yl)propanamide
N-[2-(furan-2-yl)ethyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-amine
2-(3-{[cyclohexyl(methyl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-N-ethylpyrimidin-4-amine
methyl 2-{[3-(naphthalen-1-ylmethyl)-4,5-dihydro-1,2-oxazol-5-yl]formamido}acetate
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-3-(pyridin-3-yl)propanamide
(2S,3R)-1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-methyl-2-(methylamino)pentan-1-one
1-[3-(1-benzyl-1H-pyrazol-4-yl)-4-(morpholin-4-yl)phenyl]ethan-1-one
N-{[2-(azepan-1-yl)-7-chloroquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-5-carboxamide
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-methoxy-N-methylbenzamide
(4aS,7aR)-1-[2-(3,4-dimethylphenyl)acetyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-methylacetamide
2-(2-{[(dimethyl-1,2-oxazol-4-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
3-(2-methylpropyl)-6-(oxan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
1-[(2-ethoxyphenyl)methyl]-3-(2-methoxyethyl)piperidine
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-(furan-3-ylmethyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-benzyl-3-methyl-N-[(6-methylpyridin-2-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
3-methyl-1-(2-methylphenyl)-4-[3-(propan-2-yl)-1,2-oxazol-5-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl 3-[2-(4-methoxyphenyl)acetyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(4-chlorophenyl)methyl]-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-4-(2-methylphenyl)piperazine
1-{[(3R,4R)-4-(hydroxymethyl)-1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methyl}piperidin-4-ol
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N,N-bis(prop-2-en-1-yl)benzamide
[3-({1-[2-(morpholin-4-yl)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-(piperidine-1-carbonyl)pyrazine
2-(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
3-[4-({[(2S)-1-hydroxypropan-2-yl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
N-butyl-N-[(2-fluorophenyl)methyl]-3-(5-methyl-1H-pyrazol-1-yl)propanamide
1-[1'-(3,4-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
6-[(2,3-dimethoxyphenyl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
5-(3-acetylphenoxymethyl)-N-(3,3-dimethylbutyl)-1H-pyrazole-3-carboxamide
benzyl(methyl)({3-[2-(2-methylpropyl)morpholine-4-carbonyl]-1,2-oxazol-5-yl}methyl)amine