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N-(furan-2-ylmethyl)-N,1-dimethyl-5-({[3-(trifluoromethyl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{4-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-4-oxobutyl}piperidin-2-one
1-ethyl-3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}-1H-pyrrolo[2,3-c]pyridine-5-carboxylic acid
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-[3-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
4-(5-methylpyrazine-2-carbonyl)-2-(3-phenylpropyl)morpholine
5-(3-fluorophenoxymethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
1-(2-amino-4-{[2-(dimethylamino)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-(cyclopent-2-en-1-yl)ethan-1-one
3-(isoquinolin-5-yl)-4H-chromen-4-one
(oxolan-2-ylmethyl)({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})propylamine
2-[(3,5-difluorophenyl)methyl]-8-propanoyl-2,8-diazaspiro[4.5]decan-3-one
1-[4-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
N-[4-(1,3-thiazol-4-yl)phenyl]-1-(thiophene-2-carbonyl)piperidine-3-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methoxy-2-methylpropan-1-one
1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]-2-(1,3-thiazol-2-yl)piperidine
3-({2-[1-(2-chloro-6-fluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-({7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
2-{[(1-methyl-1H-pyrazol-4-yl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amino}ethan-1-ol
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(2,3-dimethoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(furan-2-carbonyl)piperidin-4-yl]oxolane-3-carboxamide
4-{3-ethyl-5-[2-(4-methylpiperazin-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(pyridin-2-yl)acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[2-(1H-indol-1-yl)ethyl]amino}piperidin-1-yl)benzamide
1-{1-[1-(4-methylquinazolin-2-yl)pyrrolidine-2-carbonyl]piperidin-4-yl}-2-phenylethan-1-ol
(1S,6R)-9-[3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propanoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]benzoic acid
(4aS,7aR)-N-(3-cyanophenyl)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidine-3-carboxylate
(2E)-N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-4-yl)prop-2-enamide
7-methyl-3-(1,4-oxazepan-4-ylmethyl)-1,2-dihydroquinolin-2-one
3-phenoxy-N-{1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
1-(2-{4-[(2,4-dimethoxy-3-methylphenyl)methyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
(2R,6R)-1-[5-(4-chloro-2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
2-(2-chloro-4-fluorophenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
1-[(3-methyl-1H-pyrazol-5-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
3-{1-[2-(1-phenyl-1H-pyrazol-5-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-benzyl-5-(4-benzylpiperidine-1-carbonyl)-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
(1R,9S)-5-amino-3-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
2-fluoro-5-({[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]carbamoyl}amino)-N-methylbenzamide
1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-4-(pyridin-4-yl)-1,4-diazepan-6-ol
4-{[5-(5-chloro-2-fluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-1-methylpiperidine
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(isoquinoline-3-carbonyl)pyrrolidin-3-yl]methanol
3-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]-N-(2-methylphenyl)propanamide
N-(2,5-dihydroxy-2-methylpentyl)-1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
9-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-azaspiro[5.5]undecane
(4aS,7aR)-1-(1H-imidazol-2-ylmethyl)-4-[(2E)-3-phenylprop-2-en-1-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[(2,5-dimethoxyphenyl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-(cyclohex-1-en-1-ylmethyl)-3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamide