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N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}quinoxalin-2-amine
N-[2-(1H-indol-3-yl)ethyl]-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
N-(1-benzothiophen-2-ylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methylpiperidin-4-amine
N-(1,3-benzothiazol-6-yl)-4-[hydroxy(pyridin-2-yl)methyl]piperidine-1-carboxamide
1-(4-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-2-methoxyphenoxy)-3-(4-ethylpiperazin-1-yl)propan-2-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methoxyfuran-2-carboxamide
2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}acetamide
1-(6-fluoro-4-methylquinazolin-2-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
1-[(3-fluorophenyl)methyl]-5-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
1-(4-{[4-(5-propyl-1,2-oxazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
5-[2-(methylsulfanyl)phenoxymethyl]-N-[1-(pyridin-3-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
6-(2-fluoro-4-methoxyphenyl)-N,7-dimethyl-8-oxo-N-propyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
methyl 3-[2-(2-fluorophenyl)acetamido]-6-{[methyl(2-methylpropyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
(furan-2-ylmethyl)(methyl){[1-(2-methylpropyl)-2-(oxolan-2-ylmethanesulfonyl)-1H-imidazol-5-yl]methyl}amine
2-ethyl-4-methyl-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-1,3-oxazole-5-carboxamide
N-[2-(pyridin-3-yloxy)phenyl]-1-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-4-(methoxymethyl)piperidine-1-sulfonamide
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[2-(4-methoxyphenyl)ethyl]acetamide
1-[(4-ethylphenyl)methyl]-4-(2-methoxyethyl)-1,4-diazepan-5-one
4-{3-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}-3,3-dimethylpiperazin-2-one
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-4-methyl-1,2,3-thiadiazole-5-carboxamide
(1-{[1-(9H-purin-6-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
5-methoxy-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]furan-2-carboxamide
8-(1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
(3R,4R)-1-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
3-[3-(carbamoylmethyl)-1-(3-chlorophenyl)-1H-1,2,4-triazol-5-yl]-N-cyclopentylpropanamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-(2-methyl-1,3-thiazol-4-yl)-N-(2-methylpropyl)acetamide
N-({8-[(2-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-4-(piperidin-1-ylmethyl)benzamide
1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
(1S,5R)-6-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-acetamido-N-(2-methoxyphenyl)-5-[({[4-(trifluoromethyl)phenyl]methyl}amino)methyl]benzamide
5-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
4-[(1H-imidazol-2-ylmethyl)(methyl)sulfamoyl]-N-pentylbenzamide
2-acetyl-8-(3-fluoropyridin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
[(2-fluorophenyl)methyl](2-methoxyethyl){[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
benzyl (1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
1-[1-(cyclohexylmethyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(4-ethoxyphenyl)methyl]piperidin-3-yl}propanamide
5-(1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3,4-dihydro-2H-1-benzopyran-2-carboxamide
1-[3-(morpholin-4-yl)propyl]-5,5-diphenylpiperidin-2-one
6-(benzyloxy)-4-[4-(1H-pyrazol-1-yl)benzoyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
2-ethoxy-N-[(3R,4S)-4-(propan-2-yl)-1-[(trimethyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]acetamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-(1-methylpiperidin-2-yl)propanamide
5-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
N'1-[(3R,4S)-1-[(2-cyanophenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
ethyl 3-[(2-fluorophenyl)methyl]-1-[2-(1H-imidazol-1-yl)acetyl]piperidine-3-carboxylate
[5-(1H-1,3-benzodiazol-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methanamine
4-(piperidin-1-ylmethyl)-N-[1-(pyridin-3-yl)propan-2-yl]benzamide